SCHEMBL8936307

SCHEMBL8936307

BrCCC=C1c2ccccc2CCc2c1ccc1ccccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.47
CYP1A2 P05177 3/20 0.47
RET P07949 3/20 0.47
CYP2C19 P33261 2/20 0.47
SLC6A2 P23975 4/20 0.46
LMNA P02545 4/20 0.46
HTR2B P41595 3/20 0.46
HRH1 P35367 3/20 0.46
KCNH2 Q12809 3/20 0.46
ADRB2 P07550 2/20 0.46
CHRM2 P08172 2/20 0.46
CHRM4 P08173 2/20 0.46
ADRB1 P08588 2/20 0.46
HTR1A P08908 2/20 0.46
CHRM5 P08912 2/20 0.46
ADRA2A P08913 2/20 0.46
CYP2D6 P10635 2/20 0.46
CHRM1 P11229 2/20 0.46
DRD2 P14416 2/20 0.46
ADRA2B P18089 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL653565 0.83 CYP3A4 (0.63) CYP3A4CYP1A2RETCYP2C19SLC6A2
SCHEMBL6705946 0.76 BCHE (0.45) CYP1A2CYP2C19LMNAHTR1AHTT
SCHEMBL16938066 0.74 CYP3A4 (0.54) CYP3A4CYP1A2RETCYP2C19SLC6A2
SCHEMBL15908322 0.73 CYP3A4 (0.50) CYP3A4CYP1A2RETCYP2C19SLC6A2
SCHEMBL11202871 0.71 CYP3A4 (0.50) CYP3A4CYP1A2RETCYP2C19SLC6A2
SCHEMBL6962472 0.71 CYP3A4 (0.54) CYP3A4CYP1A2RETCYP2C19SLC6A2
SCHEMBL11202872 0.71 CYP3A4 (0.50) CYP3A4CYP1A2RETCYP2C19SLC6A2
SCHEMBL8936293 0.70 CYP3A4 (0.49) CYP3A4CYP1A2RETCYP2C19SLC6A2
SCHEMBL6736351 0.69 SLC6A2 (0.56) CYP3A4CYP1A2RETCYP2C19SLC6A2
SCHEMBL7815467 0.67 CYP1A2 (0.41) CYP3A4CYP1A2RETCYP2C19SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996031469-A1 N-SUBSTITUTED AZAHETEROCYCLIC CARBOXYLIC ACIDS AND ESTERS THEREOF NOVO NORDISK A/S (DK) 1996-10-10 WO disclosed