SCHEMBL8936892

SCHEMBL8936892

CC(NCC1NC(=O)NC1=O)c1ccccc1OCc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.37
TACR1 P25103 15/20 0.37
PTPN2 P17706 1/20 0.35
PTPN6 P29350 1/20 0.35
PPARG P37231 1/20 0.35
ADAM17 P78536 1/20 0.33
MLNR O43193 1/20 0.33
ABCB11 O95342 1/20 0.33
ADRB1 P08588 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
CYP2D6 P10635 1/20 0.33
CHRM1 P11229 1/20 0.33
DRD2 P14416 1/20 0.33
ADRA2C P18825 1/20 0.33
CHRM3 P20309 1/20 0.33
GLRA1 P23415 1/20 0.33
SLC6A2 P23975 1/20 0.33
HTR2C P28335 1/20 0.33
AVPR2 P30518 1/20 0.33
SLC6A4 P31645 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8936887 1.00 PTPN1 (0.37) PTPN1TACR1PTPN2PTPN6PPARG
Hydrochloric Acid SCHEMBL8936924 0.99 PTPN1 (0.36) PTPN1TACR1PTPN2PTPN6PPARG
Hydrochloric Acid SCHEMBL8936936 0.99 PTPN1 (0.36) PTPN1TACR1PTPN2PTPN6PPARG
SCHEMBL8936912 0.71 TACR1 (0.43) TACR1MLNRABCB11ADRB1ADORA3
SCHEMBL8936883 0.69 TACR1 (0.60) TACR1MLNRABCB11ADRB1ADORA3
SCHEMBL8936879 0.69 TACR1 (0.61) TACR1MLNRABCB11ADRB1ADORA3
SCHEMBL8507790 0.64 TACR1 (0.49) TACR1CYP2D6
SCHEMBL8936904 0.63 TACR1 (0.63) TACR1
SCHEMBL7704915 0.63 TACR1 (0.61) TACR1CHRM1
SCHEMBL8936871 0.63 TACR1 (0.45) TACR1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5494926-A ANTIINFLAMMATORY AGENT, ANTIARTHRITIC AGENT; TREATING PAIN, HEADACHE MERCK SHARP & DOHME LTD. (GB) 1996-02-27 US claimed
WO-1993024465-A1 2/3-(HETEROCYCLIC ALKYL AMINO)-1-(SUBST.-PHENYL-METHOXY)-ETHANES/PROPANES AS TACHYKININ-RECEPTOR ANTAGONISTS MERCK SHARP & DOHME LIMITED (GB) 1993-12-09 WO claimed