SCHEMBL8936899

SCHEMBL8936899

O=c1[nH]nc(CNC[C@@H](OCc2cc(Cl)cc(Cl)c2)c2ccccc2)[nH]1

nearest known ligand 0.52

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 14/20 0.52
CHRNB2 P17787 1/20 0.38
CHRNA4 P43681 1/20 0.38
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8936917 0.62 TACR1 (1.00) TACR1
SCHEMBL16664112 0.62 NPC1 (0.56) CHRNB2CHRNA4LMNA
SCHEMBL7668214 0.60 TSHR (0.52) TACR1LMNA
SCHEMBL16663928 0.59 CA1 (0.49) LMNA
SCHEMBL12474423 0.58 DAO (0.73) LMNA
SCHEMBL29125822 0.58 RAB9A (0.54)
SCHEMBL16663991 0.58 CA1 (0.49) LMNA
SCHEMBL16664061 0.58 CA1 (0.49) LMNA
SCHEMBL16664057 0.58 CA1 (0.49) LMNA
SCHEMBL29125683 0.57 TSHR (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5494926-A ANTIINFLAMMATORY AGENT, ANTIARTHRITIC AGENT; TREATING PAIN, HEADACHE MERCK SHARP & DOHME LTD. (GB) 1996-02-27 US disclosed
WO-1993024465-A1 2/3-(HETEROCYCLIC ALKYL AMINO)-1-(SUBST.-PHENYL-METHOXY)-ETHANES/PROPANES AS TACHYKININ-RECEPTOR ANTAGONISTS MERCK SHARP & DOHME LIMITED (GB) 1993-12-09 WO disclosed