SCHEMBL8938501

SCHEMBL8938501

O=C1CC=Cc2cc(OC3CCNCC3)c(Cl)cc21

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 1/20 0.40
HRH1 P35367 2/20 0.37
DDR1 Q08345 1/20 0.36
SLC6A4 P31645 3/20 0.33
HTR1A P08908 2/20 0.33
SLC6A2 P23975 2/20 0.33
NMT1 P30419 2/20 0.33
UTS2R Q9UKP6 2/20 0.32
P2RX3 P56373 1/20 0.32
MAPK14 Q16539 1/20 0.32
SLC6A3 Q01959 1/20 0.32
HTR6 P50406 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8938583 0.80 HRH3 (0.38)
SCHEMBL8938515 0.76 ROCK1 (0.46) HRH1
SCHEMBL1230464 0.72 HRH1 (0.46) MAP2K1HRH1SLC6A4HTR1ASLC6A2
SCHEMBL12316617 0.72 MAP2K1 (0.40) MAP2K1HRH1DDR1NMT1UTS2R
SCHEMBL12316544 0.70 MAP2K1 (0.41) MAP2K1HRH1DDR1SLC6A4HTR1A
SCHEMBL2553714 0.68 MAP2K1 (0.46) MAP2K1HRH1DDR1SLC6A4HTR1A
Hydrochloric Acid SCHEMBL15391767 0.67 MAP2K1 (0.45) MAP2K1HRH1DDR1SLC6A4HTR1A
SCHEMBL1231225 0.66 HTR2C (0.48) MAP2K1HRH1SLC6A4HTR1ASLC6A2
SCHEMBL5372606 0.65 HTR2C (0.55) SLC6A4HTR1ASLC6A2HTR6HTR2C
SCHEMBL1782182 0.65 HTR2C (0.55) SLC6A4NMT1HTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188117-B2 Piperidinyl-substituted isoquinolone derivatives SANOFI-AVENTIS (FR) 2012-05-29 US disclosed