SCHEMBL8938583

SCHEMBL8938583

CC(C)N1CCC(Oc2cc3c(cc2Cl)C(=O)CC=C3)CC1

nearest known ligand 0.38

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 18/20 0.38
CYP2D6 P10635 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8938501 0.80 MAP2K1 (0.40)
SCHEMBL8939215 0.70 HRH3 (0.38) HRH3CYP2D6
SCHEMBL5865374 0.68 HRH3 (0.47) HRH3
SCHEMBL2570202 0.67 MAP2K1 (0.62) HRH3CYP2D6
SCHEMBL5865157 0.66 SCD (0.48) HRH3CYP2D6
Hydrochloric Acid SCHEMBL1397945 0.65 HRH3 (0.53) HRH3
SCHEMBL3639284 0.63 HRH3 (0.42) HRH3
SCHEMBL8934714 0.63 HRH3 (0.39) HRH3CYP2D6
SCHEMBL19575433 0.62 HRH3 (0.41) HRH3
SCHEMBL1397997 0.62 HRH3 (0.50) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188117-B2 Piperidinyl-substituted isoquinolone derivatives SANOFI-AVENTIS (FR) 2012-05-29 US disclosed