SCHEMBL8938555

SCHEMBL8938555

COc1cc2c(=O)[nH]ccc2cc1OC1CCCCC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 8/20 0.58
MAP2K1 Q02750 1/20 0.51
ROCK2 O75116 2/20 0.47
PRKCD Q05655 2/20 0.47
PRKACA P17612 1/20 0.47
PRKG1 Q13976 1/20 0.47
PKN1 Q16512 1/20 0.47
PKN2 Q16513 1/20 0.47
AAK1 Q2M2I8 1/20 0.47
CDC42BPA Q5VT25 1/20 0.47
Q6ZSR9 Q6ZSR9 1/20 0.47
BMP2K Q9NSY1 1/20 0.47
CDC42BPB Q9Y5S2 1/20 0.47
PRKX P51817 1/20 0.46
PRKCE Q02156 1/20 0.46
PRKD1 Q15139 1/20 0.46
PDE4B Q07343 9/20 0.44
PDE4A P27815 6/20 0.44
PDE4C Q08493 6/20 0.44
PDE4D Q08499 6/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8934391 0.89 MAP2K1 (0.62) ROCK1MAP2K1ROCK2PRKCDPRKACA
SCHEMBL8934478 0.86 ROCK1 (0.49) ROCK1MAP2K1ROCK2PRKCDPRKACA
SCHEMBL8936423 0.86 ACHE (0.46) ROCK1MAP2K1ROCK2BMP2KPDE4B
SCHEMBL8938640 0.86 ROCK1 (0.76) ROCK1MAP2K1ROCK2PRKCDPRKACA
SCHEMBL8939200 0.84 ROCK1 (0.57) ROCK1MAP2K1ROCK2PRKCDPRKACA
SCHEMBL3951034 0.83 ROCK1 (0.46) ROCK1MAP2K1ROCK2PRKCDPRKACA
SCHEMBL18536013 0.83 MAP2K1 (0.72) ROCK1MAP2K1ROCK2PRKCDPRKACA
SCHEMBL8938589 0.83 ROCK1 (0.56) ROCK1MAP2K1ROCK2PRKCDPRKACA
SCHEMBL8938588 0.83 ROCK1 (0.56) ROCK1MAP2K1ROCK2PRKCDPRKACA
SCHEMBL8938521 0.80 ROCK1 (0.53) ROCK1MAP2K1ROCK2PRKCDPRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188117-B2 Piperidinyl-substituted isoquinolone derivatives SANOFI-AVENTIS (FR) 2012-05-29 US disclosed