SCHEMBL8938735

SCHEMBL8938735

CC(F)(F)c1ccc(CN2CCC(Oc3cc4cc[nH]c(=O)c4cc3Cl)CC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 2/20 0.52
ENPP2 Q13822 2/20 0.40
ROCK1 Q13464 1/20 0.40
SCN1A P35498 1/20 0.40
SCN8A Q9UQD0 1/20 0.40
ROCK2 O75116 1/20 0.38
SCD O00767 1/20 0.38
PRKACA P17612 3/20 0.37
PRKACG P22612 3/20 0.37
PRKACB P22694 3/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
ADRB2 P07550 1/20 0.37
ACHE P22303 1/20 0.37
MCHR1 Q99705 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8935011 0.93 MAP2K1 (0.54) MAP2K1ENPP2ROCK1SCN1ASCN8A
SCHEMBL8939149 0.91 ROCK1 (0.51) MAP2K1ENPP2ROCK1SCN1ASCN8A
SCHEMBL8938731 0.88 MAP2K1 (0.49) MAP2K1ENPP2ROCK1SCN1ASCN8A
SCHEMBL8935003 0.88 MAP2K1 (0.57) MAP2K1ROCK1SCN1ASCN8AROCK2
SCHEMBL8938150 0.88 MAP2K1 (0.57) MAP2K1ENPP2ROCK1ROCK2PRKACA
SCHEMBL8938278 0.88 MAP2K1 (0.59) MAP2K1ROCK1SCN1ASCN8AROCK2
SCHEMBL8938176 0.86 MAP2K1 (0.55) MAP2K1ROCK1SCN1ASCN8AROCK2
SCHEMBL8938170 0.86 MAP2K1 (0.55) MAP2K1ENPP2ROCK1ROCK2PRKACA
SCHEMBL8935032 0.86 MAP2K1 (0.51) MAP2K1ENPP2SCN1ASCN8A
SCHEMBL8934981 0.86 MAP2K1 (0.59) MAP2K1ROCK1SCN1ASCN8AROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188117-B2 Piperidinyl-substituted isoquinolone derivatives SANOFI-AVENTIS (FR) 2012-05-29 US disclosed