SCHEMBL8939149

SCHEMBL8939149

Cc1cc2c(=O)[nH]ccc2cc1OC1CCN(Cc2ccc(C(C)(F)F)cc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.51
MAP2K1 Q02750 1/20 0.41
ENPP2 Q13822 2/20 0.40
SCN1A P35498 2/20 0.38
SCN8A Q9UQD0 2/20 0.38
MCHR1 Q99705 1/20 0.38
PRKACA P17612 3/20 0.37
PRKACG P22612 3/20 0.37
PRKACB P22694 3/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
ADRB2 P07550 1/20 0.37
ACHE P22303 1/20 0.37
HTR1D P28221 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8937960 0.94 ROCK1 (0.52) ROCK1MAP2K1ENPP2ADRB2ACHE
SCHEMBL8938735 0.91 MAP2K1 (0.52) ROCK1MAP2K1ENPP2SCN1ASCN8A
SCHEMBL8937943 0.89 ROCK1 (0.56) ROCK1MAP2K1ENPP2SCN1ASCN8A
SCHEMBL8939121 0.88 ROCK1 (0.48) ROCK1MAP2K1ENPP2SCN1ASCN8A
SCHEMBL8937994 0.88 ROCK1 (0.55) ROCK1MAP2K1MCHR1PRKACAPRKACG
SCHEMBL8937905 0.87 ROCK1 (0.48) ROCK1MAP2K1ENPP2SCN1ASCN8A
SCHEMBL8937945 0.87 ROCK1 (0.56) ROCK1MAP2K1SCN1ASCN8APRKACA
SCHEMBL13890346 0.86 ROCK1 (0.53) ROCK1MAP2K1SCN1ASCN8APRKACA
SCHEMBL8938736 0.85 ROCK1 (0.53) ROCK1PRKACAMAOAMAOBADRB2
SCHEMBL8937933 0.85 ROCK1 (0.54) ROCK1MAP2K1SCN1ASCN8APRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188117-B2 Piperidinyl-substituted isoquinolone derivatives SANOFI-AVENTIS (FR) 2012-05-29 US disclosed