SCHEMBL8939121

SCHEMBL8939121

Cc1cc2c(=O)[nH]ccc2cc1OC1CCN(Cc2ccc(S(=O)(=O)C(C)(F)F)cc2)CC1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.48
ENPP2 Q13822 3/20 0.40
SCN1A P35498 7/20 0.40
SCN8A Q9UQD0 7/20 0.40
MAP2K1 Q02750 1/20 0.39
HRH1 P35367 2/20 0.37
CCR3 P51677 2/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8937905 0.94 ROCK1 (0.48) ROCK1ENPP2SCN1ASCN8AMAP2K1
SCHEMBL8938731 0.92 MAP2K1 (0.49) ROCK1ENPP2SCN1ASCN8AMAP2K1
SCHEMBL8937809 0.89 ROCK1 (0.52) ROCK1SCN1ASCN8AMAP2K1HRH1
SCHEMBL8939149 0.88 ROCK1 (0.51) ROCK1ENPP2SCN1ASCN8AMAP2K1
SCHEMBL8937960 0.87 ROCK1 (0.52) ROCK1ENPP2MAP2K1
SCHEMBL8937943 0.86 ROCK1 (0.56) ROCK1ENPP2SCN1ASCN8AMAP2K1
SCHEMBL8937994 0.85 ROCK1 (0.55) ROCK1MAP2K1HRH1CCR3KCNH2
SCHEMBL8935032 0.84 MAP2K1 (0.51) ENPP2SCN1ASCN8AMAP2K1
SCHEMBL8937945 0.84 ROCK1 (0.56) ROCK1SCN1ASCN8AMAP2K1
SCHEMBL13890346 0.83 ROCK1 (0.53) ROCK1SCN1ASCN8AMAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188117-B2 Piperidinyl-substituted isoquinolone derivatives SANOFI-AVENTIS (FR) 2012-05-29 US disclosed