SCHEMBL8939774

SCHEMBL8939774

[c]1ccc2c(c1CCCCc1ccccc1)OCO2

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.43
MAOA P21397 3/20 0.43
HTR1A P08908 1/20 0.39
SIGMAR1 Q99720 5/20 0.37
TRPA1 O75762 1/20 0.36
CCR3 P51677 1/20 0.36
POLB P06746 1/20 0.36
LTA4H P09960 1/20 0.35
CALM1 P0DP23 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8925096 0.84 ABCG2 (0.38) MAOBMAOAHTR1ACALM1
SCHEMBL6886568 0.82 AOC3 (0.34)
SCHEMBL7462090 0.81 CYP3A4 (0.33)
SCHEMBL63619 0.73 AOC3 (0.35)
SCHEMBL6570928 0.66 HTR2A (0.42) MAOBMAOASIGMAR1
SCHEMBL161183 0.66 ABCG2 (0.39)
SCHEMBL8939757 0.65 MAOA (0.42) MAOBMAOASIGMAR1
SCHEMBL3404505 0.64 ABCG2 (0.37)
SCHEMBL451456 0.64 MAOA (0.74) MAOBMAOASIGMAR1
SCHEMBL7421641 0.64 HTR2A (0.40) MAOAHTR1ASIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516797-A SUPPRESSING GRAFT REJECTION VERTEX PHARMACEUTICALS, INCORPORATED (US) 1996-05-14 US disclosed
US-5330993-A Immunosuppressive compounds VERTEX PHARMACEUTICALS, INC. (US) 1994-07-19 US disclosed