SCHEMBL8942012

SCHEMBL8942012

NCCc1ccc(NC2CN(c3c(F)cc4cc5c(=O)c(C(=O)O)cn(C6CC6)c5nc4c3F)C2)cc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 6/20 0.46
CHRM2 P08172 2/20 0.43
DRD1 P21728 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ABCC4 O15439 1/20 0.43
LMNA P02545 1/20 0.43
HSD17B10 Q99714 1/20 0.43
KCNH2 Q12809 3/20 0.41
GSK3B P49841 4/20 0.40
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
CHRM1 P11229 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
TOP2A P11388 1/20 0.38
TOP2B Q02880 1/20 0.38
DHFR P00374 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8942091 0.89 KDM4E (0.38) DPP4CHRM2DRD1KDM4ELMNA
SCHEMBL8942266 0.89 KDM4E (0.42) DPP4KDM4ELMNAHSD17B10ALDH1A1
SCHEMBL8942326 0.88 TOP1 (0.37) DPP4CHRM2DRD1KDM4EABCC4
SCHEMBL8942072 0.86 DPP4 (0.45) DPP4CHRM2DRD1KDM4EABCC4
SCHEMBL8941979 0.84 DPP4 (0.50) DPP4CHRM2DRD1KDM4EABCC4
SCHEMBL8942390 0.83 DPP4 (0.47) DPP4CHRM2DRD1KDM4EABCC4
SCHEMBL8942162 0.82 DPP4 (0.56) DPP4CHRM2DRD1KDM4EABCC4
SCHEMBL8942227 0.82 DPP4 (0.47) DPP4CHRM2DRD1KDM4EABCC4
Water SCHEMBL8942213 0.81 DPP4 (0.55) DPP4CHRM2DRD1KDM4EABCC4
SCHEMBL8942245 0.77 DPP4 (0.49) DPP4CHRM2DRD1KDM4EABCC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5556861-A 1,8 benzonaphthyridine derivatives and antimicrobial compositions LABORATOIRE ROGER BELLON (FR) 1996-09-17 US disclosed