SCHEMBL8942072

SCHEMBL8942072

NCCc1ccc(NC2CN(c3cc4nc5c(cc4cc3F)c(=O)c(C(=O)O)cn5C3CC3)C2)cc1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 6/20 0.45
CHRM2 P08172 1/20 0.44
DRD1 P21728 1/20 0.44
KDM4E B2RXH2 4/20 0.43
LMNA P02545 3/20 0.43
HSD17B10 Q99714 3/20 0.43
ABCC4 O15439 1/20 0.43
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
ALDH1A1 P00352 3/20 0.42
HPGD P15428 2/20 0.42
MAPT P10636 1/20 0.42
TOP1 P11387 1/20 0.41
CYP1A2 P05177 1/20 0.40
TOP2A P11388 1/20 0.40
CYP2C9 P11712 1/20 0.40
TOP2B Q02880 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8942049 0.89 TOP1 (0.40) KDM4ELMNAHSD17B10CA1CA2
SCHEMBL8941970 0.89 TOP1 (0.42) KDM4ELMNAHSD17B10ALDH1A1HPGD
SCHEMBL8942239 0.88 ENPP2 (0.45) KDM4ELMNAHSD17B10ALDH1A1HPGD
SCHEMBL8941918 0.88 TOP1 (0.41) KDM4ELMNAHSD17B10CA1CA2
SCHEMBL8942101 0.87 TOP1 (0.39) KDM4ELMNAHSD17B10CA1CA2
SCHEMBL8942012 0.86 DPP4 (0.46) DPP4CHRM2DRD1KDM4ELMNA
SCHEMBL7237402 0.85 DPP4 (0.49) DPP4KDM4ELMNAHSD17B10CA1
SCHEMBL8942094 0.85 DPP4 (0.48) DPP4CHRM2DRD1KDM4ELMNA
SCHEMBL8941960 0.84 DPP4 (0.49) DPP4CHRM2DRD1KDM4ELMNA
SCHEMBL8941991 0.83 DPP4 (0.48) DPP4CHRM2DRD1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5556861-A 1,8 benzonaphthyridine derivatives and antimicrobial compositions LABORATOIRE ROGER BELLON (FR) 1996-09-17 US disclosed