SCHEMBL8945814

SCHEMBL8945814

CC1=Nc2ccccc2CC(c2cccs2)N1Cc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.44
TP53 P04637 1/20 0.44
ALOX15 P16050 1/20 0.44
GSK3B P49841 1/20 0.38
POLB P06746 1/20 0.37
BCHE P06276 1/20 0.37
KMT2A Q03164 4/20 0.36
KDM4E B2RXH2 5/20 0.36
MEN1 O00255 3/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
ALDH1A1 P00352 4/20 0.35
LMNA P02545 2/20 0.35
HTT P42858 2/20 0.35
HPGD P15428 1/20 0.35
MAPT P10636 2/20 0.35
GLA P06280 1/20 0.35
ATM Q13315 1/20 0.35
MITF O75030 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8946110 0.87 GAA (0.42) GAATP53ALOX15GSK3BPOLB
SCHEMBL11271532 0.84 MEN1 (0.36) KMT2AMEN1
Hydrochloric Acid SCHEMBL11153874 0.83 MEN1 (0.36) KMT2AMEN1
SCHEMBL8945774 0.81 SLC6A2 (0.40) GAAPOLBBCHEKMT2AKDM4E
SCHEMBL8945788 0.73 MEN1 (0.38) GAAPOLBBCHEKMT2AKDM4E
Hydrochloric Acid SCHEMBL8946092 0.72 MEN1 (0.37) GAAPOLBBCHEKMT2AKDM4E
SCHEMBL8945770 0.71 SLC6A2 (0.36) GAAPOLBBCHEKMT2AKDM4E
SCHEMBL8946091 0.71 SLC6A2 (0.38) GAAPOLBBCHEKMT2AKDM4E
Hydrochloric Acid SCHEMBL8945853 0.71 SLC6A2 (0.36) GAAPOLBBCHEKMT2AKDM4E
SCHEMBL11278142 0.70 MEN1 (0.38) KMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed