SCHEMBL8946091

SCHEMBL8946091

CC(C)C1=Nc2ccccc2CC(c2cccs2)N1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
POLB P06746 1/20 0.36
BCHE P06276 2/20 0.36
NOS3 P29474 1/20 0.35
NOS2 P35228 1/20 0.35
KDM4E B2RXH2 5/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
PKM P14618 1/20 0.35
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
ALDH1A1 P00352 4/20 0.34
LMNA P02545 2/20 0.34
HPGD P15428 2/20 0.34
HTT P42858 1/20 0.34
GLA P06280 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8945737 0.99 SLC6A2 (0.37) SLC6A2SLC6A4SLC6A3POLBBCHE
SCHEMBL8945774 0.83 SLC6A2 (0.40) SLC6A2SLC6A4SLC6A3POLBBCHE
SCHEMBL8946006 0.81 HTT (0.32) KDM4EMEN1KMT2AALDH1A1HPGD
SCHEMBL8945788 0.80 MEN1 (0.38) SLC6A2SLC6A4SLC6A3POLBBCHE
Hydrochloric Acid SCHEMBL8945964 0.80 HTT (0.32) KDM4EHTTHSD17B10
Hydrochloric Acid SCHEMBL8946092 0.79 MEN1 (0.37) SLC6A2SLC6A4SLC6A3POLBBCHE
SCHEMBL8945925 0.79 ADORA2B (0.32) HRH4
SCHEMBL8945770 0.78 SLC6A2 (0.36) SLC6A2SLC6A4SLC6A3POLBBCHE
Hydrochloric Acid SCHEMBL8945853 0.77 SLC6A2 (0.36) SLC6A2SLC6A4SLC6A3POLBBCHE
Hydrochloric Acid SCHEMBL8945951 0.77 ADORA2B (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US claimed
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed