SCHEMBL8946036

SCHEMBL8946036

Cc1cn(N(CCO)c2ccncc2F)c2ccccc12

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BCHE P06276 4/20 0.54
SLC6A2 P23975 8/20 0.53
CYP2D6 P10635 1/20 0.34
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
ACHE P22303 1/20 0.31
MAOA P21397 3/20 0.30
MAOB P27338 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nerispirdine SCHEMBL29379158 0.90 SLC6A2 (0.67) BCHESLC6A2CYP2D6
Nerispirdine SCHEMBL3842518 0.90 SLC6A2 (0.67) BCHESLC6A2CYP2D6
Nerispirdine SCHEMBL3855895 0.89 SLC6A2 (0.65) BCHESLC6A2CYP2D6
SCHEMBL7614150 0.84 SLC6A2 (0.50) BCHESLC6A2CYP2D6ACHEMAOA
Hydrochloric Acid SCHEMBL7609627 0.83 SLC6A2 (0.49) BCHESLC6A2CYP2D6
SCHEMBL7611577 0.83 SLC6A2 (0.49) BCHESLC6A2CYP2D6
Hydrochloric Acid SCHEMBL7613979 0.82 SLC6A2 (0.48) BCHESLC6A2CYP2D6
SCHEMBL8946157 0.82 BCHE (0.55) BCHESLC6A2MEN1KMT2A
SCHEMBL8442522 0.79 SLC6A2 (0.71) BCHESLC6A2CYP2D6
SCHEMBL8946156 0.78 SLC6A2 (0.49) BCHESLC6A2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276156-A Antidepressants, treatment of Alzheimer*s disease HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1994-01-04 US claimed
EP-0509400-B1 1-(Pyrido[3,4-b]-1,4-oxazinyl-4-yl)-1H-indoles, intermediates and a process for their preparation, and their use as medicaments HOECHST ROUSSEL PHARMA (US) 1996-07-03 EP disclosed
US-5519131-A CYCLIZATION OF HYDROXYALKYLAMINO COMPOUND IN THE PRESENCE OF STRONG BASE SUCH AS SODIUM HYDRIDE OR POTASSIUM TERT-BUTOXIDE HOECHST MARION ROUSSEL INC. (US) 1996-05-21 US disclosed
US-5276156-A Antidepressants, treatment of Alzheimer*s disease HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1994-01-04 US disclosed
US-5214038-A Cholinesterase inhibitors, antidepressants, cognition activators HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1993-05-25 US disclosed
EP-0509400-A1 1-(Pyrido[3,4-b]-1,4-oxazinyl-4-yl)-1H-indoles, intermediates and a process for their preparation, and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-10-21 EP disclosed