SCHEMBL8946128

SCHEMBL8946128

CNC(Cc1cc(OC)ccc1N)c1sccc1C

nearest known ligand 0.70

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.35
ALDH1A1 P00352 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8946175 0.90 MEN1 (0.34) ALDH1A1CYP2D6
SCHEMBL8945809 0.85 TDP1 (0.33) ALDH1A1CYP3A4
SCHEMBL8946130 0.82 SLC6A2 (0.32)
SCHEMBL8946019 0.82 MEN1 (0.32) ALDH1A1
SCHEMBL9425401 0.82 MAPT (0.30)
SCHEMBL8945970 0.82 CYP3A4 (0.35) ALDH1A1CYP3A4
SCHEMBL8946017 0.79 ALOX5 (0.33) ALDH1A1CYP3A4
Hydrochloric Acid SCHEMBL8946060 0.79 HTR2A (0.32) HTR2AALDH1A1
SCHEMBL8946076 0.77 TDP1 (0.35) ALDH1A1CYP3A4
SCHEMBL8946111 0.76 CYP3A4 (0.39) HTR2AALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510346-A ANTIDEPRESSANTS, ANTIANXIETY AGENTS HOECHST MARION ROUSSEL, INC. (US) 1996-04-23 US disclosed
US-5292760-A 4-heteroaryl-1,3-benzodiazepines and 2-substituted-α-(heteroaryl)benzeneethanamines HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-08 US disclosed
EP-0322582-A2 4-Heteroaryl-1,3-Benzodiazepines and 2-substituted-alpha-(heteroaryl)benzeneethanamines, a process for their preparation and their use us medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-07-05 EP disclosed