SCHEMBL8946447

SCHEMBL8946447

O=C(O)c1cnc(N2CCCC2)nc1-c1ccccc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
PTPN11 Q06124 1/20 0.49
CNR2 P34972 1/20 0.48
CNR1 P21554 2/20 0.46
MAPK8 P45983 1/20 0.45
CDC7 O00311 1/20 0.45
POLB P06746 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ABCB1 P08183 1/20 0.41
LMNA P02545 1/20 0.41
CASP1 P29466 1/20 0.41
GBA1 P04062 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8946719 0.99 ALDH1A1 (0.53) ALDH1A1PTPN11CNR2CNR1MAPK8
SCHEMBL4120279 0.89 ALDH1A1 (0.45) ALDH1A1PTPN11KDM4EMEN1MAPT
SCHEMBL2954462 0.89 PTPN11 (0.52) ALDH1A1PTPN11CNR2POLBSMN1; SMN2
SCHEMBL4112070 0.89 HRH4 (0.49) ALDH1A1PTPN11CNR2KDM4EMAPT
Piperazine SCHEMBL6016442 0.88 ALDH1A1 (0.44) ALDH1A1PTPN11KDM4EMEN1MAPT
Methylpiperazine SCHEMBL6016601 0.84 HRH4 (0.44) ALDH1A1PTPN11CNR2KDM4EMAPT
Morpholine SCHEMBL6016373 0.84 PIK3CA (0.47) ALDH1A1PTPN11CNR2POLBSMN1; SMN2
SCHEMBL6016426 0.82 PTPN11 (0.53) ALDH1A1PTPN11CNR1MAPK8CDC7
SCHEMBL4129092 0.82 PTPN11 (0.53) ALDH1A1PTPN11CNR1KMT2A
SCHEMBL4129088 0.82 PTPN11 (0.53) ALDH1A1PTPN11CNR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5500424-A ENZYME INHIBITORS NIHON NOHYAKU CO., LTD. (JP) 1996-03-19 US disclosed
EP-0638557-A1 N-phenylpyri(mi)dine-N'-phenyl-urea derivatives, their preparation and their use as ACAT inhibitors NIHON NOHYAKU CO., LTD. (JP) 1995-02-15 EP disclosed