SCHEMBL8946591

SCHEMBL8946591

Cc1nc(-c2ccccc2)nc(-c2cccc([N+](=O)[O-])c2)c1NC(=O)NCCN(C)C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.49
POLB P06746 2/20 0.47
HTT P42858 2/20 0.47
ALDH1A1 P00352 7/20 0.47
MAPT P10636 4/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
GAA P10253 2/20 0.47
KDM4E B2RXH2 2/20 0.47
KMT2A Q03164 4/20 0.42
MEN1 O00255 3/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
ABCG2 Q9UNQ0 4/20 0.41
ABCC1 P33527 1/20 0.41
NPC1 O15118 1/20 0.41
RAD52 P43351 1/20 0.40
IRAK4 Q9NWZ3 1/20 0.40
ABCB1 P08183 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10375342 0.99 ATM (0.48) ATMPOLBHTTALDH1A1MAPT
SCHEMBL10375646 0.89 HTT (0.48) ATMPOLBHTTALDH1A1MAPT
SCHEMBL10375645 0.86 POLB (0.45) ATMPOLBHTTALDH1A1MAPT
SCHEMBL10375373 0.85 ALDH1A1 (0.51) ATMPOLBALDH1A1MAPTSMN1; SMN2
SCHEMBL10376290 0.84 ALDH1A1 (0.48) ATMPOLBALDH1A1MAPTSMN1; SMN2
SCHEMBL8946649 0.84 ATM (0.49) ATMPOLBHTTALDH1A1MAPT
Fumaric Acid SCHEMBL10375257 0.81 ALDH1A1 (0.49) ATMPOLBALDH1A1MAPTSMN1; SMN2
Fumaric Acid SCHEMBL10375258 0.81 ALDH1A1 (0.49) ATMPOLBALDH1A1MAPTSMN1; SMN2
SCHEMBL10376593 0.80 ALDH1A1 (0.52) POLBHTTALDH1A1MAPTSMN1; SMN2
SCHEMBL10376555 0.79 MAPT (0.45) ATMPOLBHTTALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5500424-A ENZYME INHIBITORS NIHON NOHYAKU CO., LTD. (JP) 1996-03-19 US disclosed
EP-0638557-A1 N-phenylpyri(mi)dine-N'-phenyl-urea derivatives, their preparation and their use as ACAT inhibitors NIHON NOHYAKU CO., LTD. (JP) 1995-02-15 EP disclosed