SCHEMBL8947892

SCHEMBL8947892

CC(N)c1c(-c2ccccc2)c2cc(Cl)ccc2c(=O)n1C

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 9/20 0.64
TACR1 P25103 1/20 0.45
MAPK8 P45983 2/20 0.42
CA1 P00915 4/20 0.40
CA2 P00918 4/20 0.40
ROCK2 O75116 1/20 0.40
MAP4K4 O95819 1/20 0.40
LCK P06239 1/20 0.40
CSF1R P07333 1/20 0.40
PIM1 P11309 1/20 0.40
RPS6KB1 P23443 1/20 0.40
CDK2 P24941 1/20 0.40
MAPK1 P28482 1/20 0.40
EPHA2 P29317 1/20 0.40
FLT3 P36888 1/20 0.40
FRK P42685 1/20 0.40
CLK2 P49760 1/20 0.40
GSK3A P49840 1/20 0.40
GSK3B P49841 1/20 0.40
LIMK1 P53667 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8947812 0.85 DPP4 (0.48) DPP4TACR1
SCHEMBL17718404 0.83 DPP4 (0.45) DPP4
SCHEMBL8947990 0.83 TACR1 (0.47) DPP4TACR1
SCHEMBL5232770 0.78 DPP4 (1.00) DPP4TACR1KCNA5KCNH2
SCHEMBL9176574 0.76 DPP4 (0.63) DPP4TACR1MAPK8
SCHEMBL8947899 0.76 DPP4 (1.00) DPP4TACR1MAPK8CA1CA2
SCHEMBL8787724 0.75 DPP4 (0.77) DPP4TACR1MAPK8KCNA5KCNH2
SCHEMBL3621940 0.75 DPP4 (0.62) DPP4TACR1MAPK8KCNA5KCNH2
SCHEMBL8784994 0.73 DPP4 (0.73) DPP4TACR1MAPK8KCNA5KCNH2
SCHEMBL8948092 0.73 DPP4 (0.73) DPP4TACR1MAPK8KCNA5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5527811-A CALCIUM- AND SUBSTANCE P RECEPTOR-ANTAGONIST ACTIVITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-06-18 US claimed