SCHEMBL8947951

SCHEMBL8947951

Cn1c(CNC(=O)Nc2cccc(CN)c2)c(-c2ccccc2)c2cc(Cl)ccc2c1=O

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 10/20 0.61
TACR1 P25103 3/20 0.48
MAPT P10636 3/20 0.44
LMNA P02545 1/20 0.44
CCKBR P32239 1/20 0.44
MAPK8 P45983 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
THRB P10828 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8947831 0.99 DPP4 (0.60) DPP4TACR1MAPTLMNACCKBR
SCHEMBL8947984 0.91 DPP4 (0.53) DPP4TACR1MAPTLMNAMAPK8
Hydrochloric Acid SCHEMBL8947929 0.90 DPP4 (0.52) DPP4TACR1MAPTLMNAMAPK8
SCHEMBL8947968 0.90 DPP4 (0.52) DPP4TACR1MAPTLMNACCKBR
SCHEMBL8947960 0.90 DPP4 (0.52) DPP4TACR1MAPTLMNACCKBR
SCHEMBL8947887 0.90 DPP4 (0.52) DPP4TACR1MAPTLMNAMAPK8
SCHEMBL8947965 0.90 DPP4 (0.52) DPP4TACR1MAPTLMNAMAPK8
SCHEMBL8948130 0.90 DPP4 (0.52) DPP4TACR1MAPTLMNAMAPK8
Hydrochloric Acid SCHEMBL8948140 0.89 DPP4 (0.51) DPP4TACR1MAPTLMNAMAPK8
Hydrochloric Acid SCHEMBL8948054 0.89 DPP4 (0.51) DPP4TACR1MAPTLMNAMAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5527811-A CALCIUM- AND SUBSTANCE P RECEPTOR-ANTAGONIST ACTIVITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-06-18 US claimed
EP-0634402-A1 Isochinolinone derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1995-01-18 EP claimed