SCHEMBL8947887

SCHEMBL8947887

CN(C)Cc1cccc(NC(=O)NCc2c(-c3ccccc3)c3cc(Cl)ccc3c(=O)n2C)c1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 7/20 0.52
KCNA5 P22460 1/20 0.47
KCNH2 Q12809 1/20 0.47
TACR1 P25103 5/20 0.47
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
ACP1 P24666 2/20 0.43
LSS P48449 1/20 0.42
MAPK8 P45983 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8948140 0.99 DPP4 (0.51) DPP4KCNA5KCNH2TACR1LMNA
SCHEMBL8948186 0.92 DPP4 (0.50) DPP4KCNA5KCNH2TACR1LMNA
SCHEMBL8948142 0.91 LSS (0.53) DPP4KCNA5KCNH2TACR1LSS
SCHEMBL8947888 0.91 DPP4 (0.54) DPP4KCNA5KCNH2TACR1ACP1
Hydrochloric Acid SCHEMBL8948118 0.90 TACR1 (0.50) KCNA5KCNH2TACR1MAPT
SCHEMBL8948026 0.90 DPP4 (0.49) DPP4KCNA5KCNH2TACR1LMNA
SCHEMBL8947984 0.90 DPP4 (0.53) DPP4TACR1LMNAMAPTMAPK8
SCHEMBL8947951 0.90 DPP4 (0.61) DPP4TACR1LMNAMAPTMAPK8
SCHEMBL8947968 0.89 DPP4 (0.52) DPP4TACR1LMNAMAPTMAPK8
Hydrochloric Acid SCHEMBL8947929 0.89 DPP4 (0.52) DPP4TACR1LMNAMAPTMAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5527811-A CALCIUM- AND SUBSTANCE P RECEPTOR-ANTAGONIST ACTIVITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-06-18 US claimed
EP-0634402-A1 Isochinolinone derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1995-01-18 EP claimed
US-5527811-A CALCIUM- AND SUBSTANCE P RECEPTOR-ANTAGONIST ACTIVITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-06-18 US disclosed
EP-0634402-A1 Isochinolinone derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1995-01-18 EP disclosed