SCHEMBL8947993

SCHEMBL8947993

Cc1cc2c(-c3ccccc3)c(CCN)n(C)c(=O)c2cc1C

nearest known ligand 0.71

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 6/20 0.71
TACR1 P25103 13/20 0.56
KCNA5 P22460 1/20 0.47
KCNH2 Q12809 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5236388 0.89 DPP4 (0.70) DPP4TACR1KCNA5KCNH2
SCHEMBL8785566 0.86 TACR1 (0.56) DPP4TACR1KCNA5KCNH2
SCHEMBL8947816 0.86 DPP4 (0.74) DPP4TACR1KCNA5KCNH2
SCHEMBL8948096 0.84 TACR1 (0.54) DPP4TACR1KCNA5KCNH2
SCHEMBL8785003 0.83 TACR1 (0.58) DPP4TACR1KCNA5KCNH2
SCHEMBL8947899 0.83 DPP4 (1.00) DPP4TACR1KCNA5KCNH2
SCHEMBL2900202 0.81 KCNA5 (0.73) DPP4TACR1KCNA5KCNH2
SCHEMBL8784483 0.81 TACR1 (0.56) DPP4TACR1KCNA5KCNH2
Hydrochloric Acid SCHEMBL2901589 0.80 DPP4 (0.71) DPP4TACR1KCNA5KCNH2
SCHEMBL8784775 0.80 TACR1 (0.55) DPP4TACR1KCNA5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5527811-A CALCIUM- AND SUBSTANCE P RECEPTOR-ANTAGONIST ACTIVITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-06-18 US claimed