SCHEMBL8947995

SCHEMBL8947995

Cc1cccc(NC(=O)NCc2c(-c3ccccc3)c3cc(Cl)ccc3c(=O)n2C)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.56
DPP4 P27487 7/20 0.56
ALDH1A1 P00352 3/20 0.46
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
TP53 P04637 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
MAPT P10636 2/20 0.44
PLA2G1B P04054 1/20 0.44
ATG4B Q9Y4P1 1/20 0.44
MAPK8 P45983 1/20 0.44
CNR1 P21554 1/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
USP2 O75604 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
KDM4E B2RXH2 1/20 0.43
THRB P10828 1/20 0.43
TDP1 Q9NUW8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8459967 0.90 TACR1 (0.59) TACR1NPC1RAB9ASMN1; SMN2TP53
SCHEMBL8948077 0.90 DPP4 (0.55) TACR1DPP4ALDH1A1NPC1RAB9A
SCHEMBL8947972 0.89 DPP4 (0.54) TACR1DPP4ALDH1A1NPC1RAB9A
SCHEMBL8947979 0.89 DPP4 (0.54) TACR1DPP4ALDH1A1NPC1RAB9A
SCHEMBL8947941 0.89 TACR1 (0.71) TACR1NPC1RAB9ASMN1; SMN2MEN1
SCHEMBL8947829 0.88 DPP4 (0.53) TACR1DPP4ALDH1A1NPC1RAB9A
SCHEMBL8947984 0.88 DPP4 (0.53) TACR1DPP4ALDH1A1NPC1RAB9A
SCHEMBL8947951 0.88 DPP4 (0.61) TACR1DPP4ALDH1A1NPC1RAB9A
Hydrochloric Acid SCHEMBL8947929 0.88 DPP4 (0.52) TACR1DPP4ALDH1A1NPC1RAB9A
Hydrochloric Acid SCHEMBL8947831 0.88 DPP4 (0.60) TACR1DPP4ALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5527811-A CALCIUM- AND SUBSTANCE P RECEPTOR-ANTAGONIST ACTIVITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-06-18 US disclosed
EP-0634402-A1 Isochinolinone derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1995-01-18 EP disclosed