SCHEMBL8948135

SCHEMBL8948135

O=C(c1ccc(F)cc1)C1CCN(CCn2c(=O)oc3ccccc32)CC1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.57
HTR2C P28335 4/20 0.57
CYP1A2 P05177 3/20 0.57
CYP3A4 P08684 3/20 0.57
HTR1A P08908 2/20 0.57
CYP2C9 P11712 2/20 0.57
DRD2 P14416 2/20 0.57
HPGD P15428 2/20 0.57
HTR7 P34969 2/20 0.57
HTR6 P50406 2/20 0.57
MEN1 O00255 1/20 0.57
ALDH1A1 P00352 1/20 0.57
LMNA P02545 1/20 0.57
MAPT P10636 1/20 0.57
ADRA2B P18089 1/20 0.57
ADRA2C P18825 1/20 0.57
DRD1 P21728 1/20 0.57
DRD4 P21917 1/20 0.57
HTR1D P28221 1/20 0.57
HTR1B P28222 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11785003 0.94 CHRM1 (0.58) HTR2ACYP1A2CYP3A4CYP2D6KDM4E
SCHEMBL7766399 0.81 HTR2A (0.49) HTR2AHTR2CHTR7HTR6SLC6A4
SCHEMBL14318600 0.80 HTR2A (0.81) HTR2AHTR2CCYP1A2CYP3A4HTR7
SCHEMBL8947873 0.80 HTR2A (0.56) HTR2AHTR2CCYP1A2CYP3A4HTR7
SCHEMBL8948121 0.79 HTR2A (0.57) HTR2AHTR2CCYP1A2CYP3A4HTR1A
SCHEMBL8018901 0.79 HTR2A (0.78) HTR2AHTR2CCYP1A2CYP3A4HTR1A
Hydrochloric Acid SCHEMBL8025211 0.78 HTR2A (0.60) HTR2AHTR2CCYP1A2CYP3A4HTR1A
SCHEMBL12124768 0.77 DRD2 (0.75) DRD2DRD4
Hydrochloric Acid SCHEMBL8021166 0.77 HTR2A (0.61) HTR2AHTR2CCYP1A2CYP3A4HTR1A
SCHEMBL29367143 0.77 HTR2A (0.66) HTR2AHTR2CCYP1A2CYP3A4HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5534517-A (Aryl(alkyl)carbonyl)-heterocyclic compounds and their use in the treatment of anxiety and depression ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
US-5387586-A Analgesics, nervous system disorders ADIR ET COMPAGNIE (FR) 1995-02-07 US disclosed
EP-0613898-A1 Aryl or arylalkyl-carbonyl heterocyclic derivatives, processes for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1994-09-07 EP disclosed