SCHEMBL8949035

SCHEMBL8949035

CCOC(=O)c1cnc(-c2ccc(C(N)=O)cc2)[nH]c1=O

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.60
ALDH1A1 P00352 4/20 0.60
L3MBTL1 Q9Y468 4/20 0.55
CA12 O43570 4/20 0.49
CA1 P00915 4/20 0.49
CA2 P00918 4/20 0.49
CA6 P23280 4/20 0.49
CA7 P43166 4/20 0.49
CA13 Q8N1Q1 4/20 0.49
PARP1 P09874 1/20 0.49
GAA P10253 1/20 0.49
MAPT P10636 5/20 0.46
POLB P06746 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
TP53 P04637 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
LMNA P02545 2/20 0.44
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4949585 0.85 KDM4E (0.63) KDM4EALDH1A1L3MBTL1GAAMAPT
SCHEMBL2897245 0.85 KDM4E (0.72) KDM4EALDH1A1L3MBTL1GAAMAPT
SCHEMBL11628696 0.84 KDM4E (0.75) KDM4EALDH1A1L3MBTL1GAAMAPT
SCHEMBL4763787 0.84 KDM4E (0.64) KDM4EALDH1A1L3MBTL1GAAMAPT
SCHEMBL23574396 0.83 KDM4E (0.64) KDM4EALDH1A1L3MBTL1CA12CA1
SCHEMBL4376727 0.82 KDM4E (0.76) KDM4EALDH1A1L3MBTL1GAAMAPT
SCHEMBL9199571 0.81 KDM4E (0.67) KDM4EALDH1A1L3MBTL1CA12CA1
SCHEMBL8948970 0.80 KDM6B (0.44)
SCHEMBL11626689 0.76 KDM4E (0.57) KDM4EALDH1A1L3MBTL1CA12CA1
SCHEMBL11631180 0.75 KDM4E (0.54) KDM4EALDH1A1L3MBTL1CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563268-A FOR PREVENTING CELL AGGLOMERATION, TREATING THROMBOSIS, ARTERIOSCLEROSIS, BRAIN, LUNG OR CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1996-10-08 US disclosed
US-5418233-A FOR INHIBITING CELL AGGREGATION KARL THOMAE GMBH (DE) 1995-05-23 US disclosed
EP-0537696-A1 Heterobiaryl derivatives, medicines containing those compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-04-21 EP disclosed