SCHEMBL8950488

SCHEMBL8950488

O=C(O)CN1CCN(CC(=O)O)CC(=O)NCC#CC#CCNC(=O)CN(CC(=O)O)CCN(CC(=O)O)CCN(CC(=O)O)CC(=O)NCC#CC#CCNC(=O)CN(CC(=O)O)CC1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
TSHR P16473 1/20 0.34
SLC6A9 P48067 1/20 0.33
TGM2 P21980 1/20 0.32
S1PR1 P21453 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8950554 0.82 SMN1; SMN2 (0.44) HSD17B10SMN1; SMN2TSHRSLC6A9TGM2
SCHEMBL8950538 0.82 SMN1; SMN2 (0.44) HSD17B10SMN1; SMN2TSHRSLC6A9TGM2
SCHEMBL8950473 0.79 SMN1; SMN2 (0.43) HSD17B10SMN1; SMN2TSHRSLC6A9
SCHEMBL8950614 0.79 SMN1; SMN2 (0.43) HSD17B10SMN1; SMN2TSHRSLC6A9
SCHEMBL8950480 0.78 HSD17B10 (0.44) HSD17B10SMN1; SMN2TSHRSLC6A9TGM2
SCHEMBL8950521 0.78 SMN1; SMN2 (0.39) HSD17B10SMN1; SMN2TSHRSLC6A9TGM2
SCHEMBL166595 0.76 SMN1; SMN2 (0.52) HSD17B10SMN1; SMN2TSHR
SCHEMBL5590521 0.70 HSD17B10 (0.37) HSD17B10TSHRSLC6A9TGM2S1PR1
SCHEMBL273928 0.69 HSD17B10 (0.42) HSD17B10TSHRSLC6A9
Trifluoroacetic Acid SCHEMBL28509604 0.69 SMN1; SMN2 (0.46) HSD17B10SMN1; SMN2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0556240-B1 CHELATING AGENTS NYCOMED SALUTAR INC (US) 1996-07-10 EP claimed
US-5556968-A Polyazamacrocycle chelating agents with amide linkages NYCOMED SALUTAR, INC. (US) 1996-09-17 US disclosed
WO-1992008707-A1 CHELATING AGENTS COCKBAIN, JULIAN, RODERICK, MICHAELSON (GB) 1992-05-29 WO disclosed