SCHEMBL8950554

SCHEMBL8950554

O=C(O)CN1CCN(CC(=O)O)CC(=O)NCCNC(=O)CN(CC(=O)O)CCN(CC(=O)O)CCN(CC(=O)O)CC(=O)NCCNC(=O)CN(CC(=O)O)CC1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.44
HSD17B10 Q99714 1/20 0.41
TSHR P16473 2/20 0.39
SLC6A9 P48067 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
KMT2A Q03164 1/20 0.37
TOP2A P11388 1/20 0.35
TOP2B Q02880 1/20 0.35
TGM2 P21980 1/20 0.35
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
S1PR1 P21453 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8950538 1.00 SMN1; SMN2 (0.44) SMN1; SMN2HSD17B10TSHRSLC6A9L3MBTL1
SCHEMBL8950473 0.93 SMN1; SMN2 (0.43) SMN1; SMN2HSD17B10TSHRSLC6A9L3MBTL1
SCHEMBL8950614 0.93 SMN1; SMN2 (0.43) SMN1; SMN2HSD17B10TSHRSLC6A9L3MBTL1
SCHEMBL166595 0.91 SMN1; SMN2 (0.52) SMN1; SMN2HSD17B10TSHRL3MBTL1KMT2A
SCHEMBL8950480 0.85 HSD17B10 (0.44) SMN1; SMN2HSD17B10TSHRSLC6A9KMT2A
SCHEMBL8950521 0.84 SMN1; SMN2 (0.39) SMN1; SMN2HSD17B10TSHRSLC6A9L3MBTL1
SCHEMBL8950488 0.82 HSD17B10 (0.36) SMN1; SMN2HSD17B10TSHRSLC6A9TGM2
Trifluoroacetic Acid SCHEMBL28509604 0.82 SMN1; SMN2 (0.46) SMN1; SMN2HSD17B10TSHRL3MBTL1KMT2A
SCHEMBL6625231 0.81 TSHR (0.40) SMN1; SMN2HSD17B10TSHRSLC6A9TGM2
SCHEMBL15698482 0.80 CHRM5 (0.38) SMN1; SMN2HSD17B10TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5556968-A Polyazamacrocycle chelating agents with amide linkages NYCOMED SALUTAR, INC. (US) 1996-09-17 US claimed
EP-0556240-B1 CHELATING AGENTS NYCOMED SALUTAR INC (US) 1996-07-10 EP claimed
EP-0556240-A1 CHELATING AGENTS. COCKBAIN JULIAN R M (GB) 1993-08-25 EP claimed
WO-1992008707-A1 CHELATING AGENTS COCKBAIN, JULIAN, RODERICK, MICHAELSON (GB) 1992-05-29 WO claimed
US-5556968-A Polyazamacrocycle chelating agents with amide linkages NYCOMED SALUTAR, INC. (US) 1996-09-17 US disclosed
EP-0556240-B1 CHELATING AGENTS NYCOMED SALUTAR INC (US) 1996-07-10 EP disclosed
WO-1992008707-A1 CHELATING AGENTS COCKBAIN, JULIAN, RODERICK, MICHAELSON (GB) 1992-05-29 WO disclosed