SCHEMBL8952162

SCHEMBL8952162

CCCCCn1cc(C#N)c(-c2ccccc2)c1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 2/20 0.40
KDM4E B2RXH2 4/20 0.39
ALDH1A1 P00352 3/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
HPGD P15428 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MAPK1 P28482 1/20 0.37
TSHR P16473 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14288449 0.82 TLR8 (0.47) TLR8KDM4EALDH1A1CNR1CNR2
SCHEMBL14288455 0.79 TSHR (0.50) TLR8ALDH1A1CNR1CNR2L3MBTL1
SCHEMBL10503713 0.76 TSHR (0.38) KDM4EALDH1A1GLAGAAHPGD
Octane SCHEMBL9620215 0.74 ESR2 (0.53) KDM4EALDH1A1GAAHPGDL3MBTL1
Decane SCHEMBL9620442 0.74 ESR2 (0.53) KDM4EALDH1A1GAAHPGDL3MBTL1
SCHEMBL1779746 0.74 KDM4E (0.47) KDM4EALDH1A1GLAGAAHPGD
SCHEMBL3595050 0.73 STAT3 (0.49)
SCHEMBL22749023 0.72 CNR1 (0.48) ALDH1A1CNR1CNR2
SCHEMBL13404301 0.70 POLB (0.52) KDM4EALDH1A1HPGDTSHRSMN1; SMN2
SCHEMBL11552875 0.70 ALDH1A1 (0.35) KDM4EALDH1A1GLAGAACNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5514816-A REACTION OF DIFLUOROBENZO-1,3-DIOXOLE WITH METAL COMPOUNDS FOR INSECTICIDES CIBA-GEIGY CORPORATION (US) 1996-05-07 US disclosed
US-5496848-A Process for the preparation of substituted difluorobenzo-1,3-dioxoles CIBA-GEIGY CORPORATION (US) 1996-03-05 US disclosed
US-5493032-A INSECTICIDES, MICROBIOCIDES CIBA-GEIGY CORPORATION (US) 1996-02-20 US disclosed
US-5420301-A Process for the preparation of substituted difluorobenzo-1,3-dioxoles CIBA-GEIGY CORPORATION (US) 1995-05-30 US disclosed
EP-0333661-B1 Process for the preparation of a pyrole derivative CIBA GEIGY AG (CH) 1994-04-27 EP disclosed
US-5281718-A Reacting in one pot reaction 2,2-difluorobenzodioxole with an organometal compound or metal to form 4-metallo-2,2-difluorobenzodioxole, reacting with unsaturated nitrile, then with isocyanide CIBA-GEIGY CORPORATION (US) 1994-01-25 US disclosed
US-5194628-A Reacting metallo-difluorobenzodioxole with unsaturated nitrile and then with sulfonylmethyl isocyanide CIBA-GEIGY CORPORATION (US) 1993-03-16 US disclosed
EP-0333661-A2 Process for the preparation of a pyrole derivative CIBA-GEIGY AG (CH) 1989-09-20 EP disclosed