SCHEMBL8955949

SCHEMBL8955949

CC(=O)Nc1ccc(-n2nc(C(F)(F)F)cc2-c2ccc(S(C)(=O)=O)cc2)cc1

nearest known ligand 0.77

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.77
PTGS1 P23219 2/20 0.70
CYP2C9 P11712 1/20 0.70
AOC3 Q16853 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6013902 0.90 PTGS2 (0.77) PTGS2PTGS1CYP2C9
SCHEMBL19953620 0.87 PTGS2 (0.70) PTGS2PTGS1CYP2C9AOC3
SCHEMBL7243347 0.86 PTGS2 (0.81) PTGS2PTGS1CYP2C9
Hydrochloric Acid SCHEMBL9207228 0.85 PTGS2 (0.79) PTGS2PTGS1CYP2C9
SCHEMBL7457684 0.85 PTGS2 (0.74) PTGS2PTGS1CYP2C9
SCHEMBL7466325 0.84 PTGS2 (0.80) PTGS2PTGS1CYP2C9
SCHEMBL8953884 0.84 AOC3 (0.62) PTGS2PTGS1AOC3
SCHEMBL9204374 0.84 PTGS2 (0.69) PTGS2PTGS1CYP2C9
SCHEMBL8925698 0.83 PTGS2 (0.71) PTGS2PTGS1CYP2C9
SCHEMBL9208661 0.83 PTGS2 (0.71) PTGS2PTGS1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0731794-A1 1,4,5-TRIPHENYL PYRAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION AND INFLAMMATION-RELATED DISORDERS SEARLE & CO (US) 1996-09-18 EP disclosed
WO-1995015317-A1 1,4,5-TRIPHENYL PYRAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION AND INFLAMMATION-RELATED DISORDERS G.D. SEARLE & CO. (US) 1995-06-08 WO disclosed