SCHEMBL8957265

SCHEMBL8957265

COc1ccccc1N1CCN(CCl)CC1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.69
MAPK1 P28482 2/20 0.67
DRD3 P35462 3/20 0.66
HTR1A P08908 2/20 0.64
ADRA1D P25100 1/20 0.64
ADRA1A P35348 1/20 0.64
ADRA1B P35368 1/20 0.64
KDM4E B2RXH2 3/20 0.62
LMNA P02545 1/20 0.62
HTT P42858 1/20 0.62
TDP1 Q9NUW8 1/20 0.62
HTR7 P34969 2/20 0.61
KMT2A Q03164 2/20 0.61
ALDH1A1 P00352 1/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
DRD4 P21917 1/20 0.61
HRH2 P25021 1/20 0.61
HRH1 P35367 1/20 0.61
MEN1 O00255 1/20 0.60
CYP1A2 P05177 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1253155 0.87 DRD2 (0.75) DRD2MAPK1DRD3HTR1AADRA1D
SCHEMBL30206503 0.86 DRD2 (0.78) DRD2DRD3HTR1AADRA1DADRA1A
SCHEMBL1255253 0.86 DRD2 (0.78) DRD2DRD3HTR1AADRA1DADRA1A
SCHEMBL4617829 0.85 DRD2 (0.77) DRD2MAPK1DRD3HTR1AADRA1D
SCHEMBL10548333 0.84 DRD2 (0.62) DRD2MAPK1DRD3HTR1AADRA1D
Hydrochloric Acid SCHEMBL11651993 0.84 DRD2 (0.76) DRD2DRD3HTR1AADRA1DADRA1A
Hydrochloric Acid SCHEMBL8980706 0.84 DRD2 (0.76) DRD2DRD3HTR1AADRA1DADRA1A
SCHEMBL9225440 0.84 MAPK1 (0.81) DRD2MAPK1DRD3ADRA1DADRA1A
SCHEMBL12304200 0.84 DRD2 (0.66) DRD2MAPK1DRD3HTR1AADRA1D
SCHEMBL5307095 0.83 DRD2 (0.69) DRD2MAPK1DRD3HTR1AADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5539107-A REACTION OF CHLOROPYRIDINE AND CHLOROQUINOLINES WITH MERCAPTOANILINES OR BIS/O-AMINOPHENYL DISULFIDE ASTA MEDICA AKTIENGESELLSCHAFT (DE) 1996-07-23 US disclosed
US-5446148-A Chemical intermediates for making antitussive agent, antihistamines and antipsychotic agent; efficiency, by-product inhibition ASTA MEDICA AKTIENGESELLSCHAFT (DE) 1995-08-29 US disclosed
EP-0611757-A1 Process for the preparation of azaphenothiazines ASTA Medica Aktiengesellschaft (DE) 1994-08-24 EP disclosed