SCHEMBL8958503

SCHEMBL8958503

NCCN(CCN)Cc1ccc(Br)cc1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.52
HTR2A P28223 1/20 0.52
PYCR1 P32322 6/20 0.52
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
HRH3 Q9Y5N1 1/20 0.42
MAPT P10636 1/20 0.41
IDO1 P14902 2/20 0.40
MAOB P27338 1/20 0.40
CARM1 Q86X55 1/20 0.39
PRMT6 Q96LA8 1/20 0.39
PRMT8 Q9NR22 1/20 0.39
GBA1 P04062 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4406268 0.89 HRH3 (0.50) PYCR1HRH3MAPTCARM1PRMT6
SCHEMBL29083510 0.81 PYCR1 (0.64) TAAR1HTR2APYCR1KDM4EALDH1A1
SCHEMBL6268253 0.80 PYCR1 (0.53) TAAR1HTR2APYCR1KDM4EALDH1A1
SCHEMBL9125321 0.80 MAPT (0.62) ALDH1A1HRH3MAPTMAOBCARM1
SCHEMBL4592016 0.78 PYCR1 (0.52) TAAR1PYCR1KDM4EALDH1A1HRH3
SCHEMBL2346063 0.77 CARM1 (0.63) TAAR1HTR2AKDM4EALDH1A1CARM1
Hydrochloric Acid SCHEMBL3665790 0.76 CARM1 (0.61) TAAR1HTR2AKDM4EALDH1A1CARM1
SCHEMBL29860798 0.76 CARM1 (0.61) TAAR1HTR2AKDM4EALDH1A1CARM1
SCHEMBL17795575 0.75 TAAR1 (0.44) TAAR1HTR2APYCR1KDM4EALDH1A1
SCHEMBL713426 0.75 MAPT (0.55) HRH3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0540975-B1 Diethylenetriamine derivatives and their use for diagnostic and therapeutic purposes BAYER AG (DE) 1996-01-10 EP disclosed
EP-0540975-A1 Diethylenetriamine derivatives and their use for diagnostic and therapeutic purposes BAYER AG (DE) 1993-05-12 EP disclosed