SCHEMBL8959136

SCHEMBL8959136

COP(=O)(Cc1ccccc1F)OC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.42
TAAR1 Q96RJ0 3/20 0.41
LMNA P02545 4/20 0.39
ALDH1A1 P00352 4/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
HTT P42858 1/20 0.39
MAOB P27338 1/20 0.38
KDM4E B2RXH2 2/20 0.38
AOC3 Q16853 1/20 0.38
HPGD P15428 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TSHR P16473 1/20 0.37
CYP1A2 P05177 1/20 0.37
POLB P06746 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
MAPT P10636 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6575682 0.86 TSHR (0.46) LMNAALDH1A1L3MBTL1HTTHPGD
SCHEMBL9172183 0.82 HTT (0.36) LMNAL3MBTL1HTTHPGDSMN1; SMN2
SCHEMBL4538982 0.81 KCNH2 (0.43) IDO1TAAR1LMNAALDH1A1KDM4E
SCHEMBL8958927 0.78 HPGD (0.43) TAAR1LMNAALDH1A1L3MBTL1HTT
SCHEMBL6384988 0.77 IDO1 (0.42) IDO1TAAR1ALDH1A1L3MBTL1HTT
SCHEMBL8958923 0.77 IDO1 (0.42) IDO1TAAR1LMNAALDH1A1L3MBTL1
SCHEMBL11710711 0.77 TSHR (0.53) IDO1TAAR1LMNAL3MBTL1HTT
SCHEMBL9021319 0.77 TSHR (0.40) IDO1LMNAALDH1A1L3MBTL1HTT
SCHEMBL4030757 0.77 FDPS (0.43) LMNAALDH1A1L3MBTL1HTTKDM4E
SCHEMBL28479763 0.77 IDO1 (0.42) IDO1TAAR1LMNAALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5500417-A ANTIARTHRITIC THE UPJOHN COMPANY (US) 1996-03-19 US claimed
EP-0661978-A1 ARYLMETHYLPHOSPHONATES AND PHOSPHONIC ACIDS USEFUL AS ANTI-INFLAMMATORY AGENTS PHARMACIA & UPJOHN COMPANY (US) 1995-07-12 EP claimed
WO-1994007501-A1 ARYLMETHYLPHOSPHONATES AND PHOSPHONIC ACIDS USEFUL AS ANTI-INFLAMMATORY AGENTS THE UPJOHN COMPANY (US) 1994-04-14 WO claimed