SCHEMBL8959641

SCHEMBL8959641

CC(O)Cn1ccc2cc(F)c(C(C)C)cc21

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 16/20 0.56
HTR2A P28223 14/20 0.56
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51
HTR2B P41595 1/20 0.51
KDM4E B2RXH2 1/20 0.37
EIF4A3 P38919 1/20 0.35
PRMT5 O14744 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8959629 1.00 HTR2C (0.56) HTR2CHTR2ACYP1A2CYP3A4CYP2C9
SCHEMBL26674202 0.88 HTR2C (0.63) HTR2CHTR2ACYP1A2CYP3A4CYP2C9
SCHEMBL8959535 0.88 HTR2C (0.71) HTR2CHTR2ACYP1A2CYP3A4CYP2C9
SCHEMBL8959539 0.88 HTR2C (0.71) HTR2CHTR2ACYP1A2CYP3A4CYP2C9
SCHEMBL8959648 0.88 HTR2C (0.71) HTR2CHTR2ACYP1A2CYP3A4CYP2C9
SCHEMBL9233642 0.85 HTR2C (0.78) HTR2CHTR2ACYP1A2CYP3A4CYP2C9
SCHEMBL8959579 0.82 HTR2C (0.74) HTR2CHTR2ACYP1A2CYP3A4CYP2C9
SCHEMBL8959895 0.82 HTR2C (0.74) HTR2CHTR2ACYP1A2CYP3A4CYP2C9
SCHEMBL8959583 0.82 HTR2C (0.74) HTR2CHTR2ACYP1A2CYP3A4CYP2C9
SCHEMBL26674263 0.81 HTR2C (0.50) HTR2CHTR2ACYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1061341-C 1-amino-ethylindole-derivatives HOFFMANN LA ROCHE (CH) 2001-01-31 CN disclosed
US-5494928-A FOR CENTRAL NERVOUS SYSTEM DISORDERS, BLOCKING SEROTONIN RECEPTORS, ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed