Epidepride

Epidepride

SCHEMBL8961795

CCN1CCC[C@H]1CNC(=O)c1cc(I)cc(OC)c1OC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.81
DRD3 P35462 3/20 0.80
DRD4 P21917 1/20 0.80
ABCG2 Q9UNQ0 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Epidepride SCHEMBL29521228 1.00 DRD2 (0.81) DRD2DRD3DRD4ABCG2
Epidepride SCHEMBL8961800 1.00 DRD2 (0.81) DRD2DRD3DRD4ABCG2
SCHEMBL27678962 0.89 DRD2 (1.00) DRD2DRD3DRD4ABCG2
SCHEMBL10355427 0.88 DRD2 (0.80) DRD2DRD3ABCG2
SCHEMBL10355426 0.88 DRD2 (0.80) DRD2DRD3ABCG2
SCHEMBL10355398 0.87 DRD2 (0.81) DRD2DRD3ABCG2
SCHEMBL5477770 0.87 DRD3 (1.00) DRD2DRD3DRD4ABCG2
SCHEMBL10355400 0.87 DRD2 (0.81) DRD2DRD3ABCG2
SCHEMBL10355469 0.87 DRD3 (1.00) DRD2DRD3DRD4ABCG2
SCHEMBL10355399 0.87 DRD2 (0.81) DRD2DRD3ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092243-B1 IONIC LIQUID SUPPORTED ORGANOTIN REAGENTS FOR THE MANUFACTURING OF RADIOPHARMACEUTICALS COMPOUNDS CENTRE NAT RECH SCIENT (FR) 2019-06-19 EP disclosed
US-5480631-A Radioiodinated benzamines and method of their use as radioimaging VANDERBILT UNIVERSITY (US) 1996-01-02 US disclosed
EP-0207913-A1 Catechol carboxamides, process for their preparation, intermediates and a pharmaceutical preparation Astra Läkemedel Aktiebolag (SE) 1987-01-07 EP disclosed
WO-1986007591-A1 CATECHOLCARBOXAMIDES, PROCESS FOR THEIR PREPARATION, INTERMEDIATES AND A PHARMACEUTICAL PREPARATION Astra Läkemedel Aktiebolag (SE) 1986-12-31 WO disclosed