SCHEMBL8962138

SCHEMBL8962138

CC(C)(C)c1cc(/C=C2/SC(=O)NC2=O)cc(C(C)(C)C)c1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 1.00
PTGS1 P23219 4/20 1.00
NAT1 P18440 1/20 0.67
CISD1 Q9NZ45 1/20 0.62
MAOA P21397 1/20 0.62
MAOB P27338 1/20 0.62
IGF1R P08069 2/20 0.62
AKR1B1 P15121 1/20 0.58
HPGD P15428 1/20 0.58
GSK3B P49841 1/20 0.58
RAB9A P51151 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
GAA P10253 1/20 0.57
ALOX5 P09917 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3667218 1.00 PTGS2 (1.00) PTGS2PTGS1NAT1CISD1MAOA
SCHEMBL3667216 1.00 PTGS2 (1.00) PTGS2PTGS1NAT1CISD1MAOA
Choline SCHEMBL7698143 0.88 PTGS2 (0.77) PTGS2PTGS1NAT1CISD1MAOA
Choline SCHEMBL7698141 0.88 PTGS2 (0.77) PTGS2PTGS1NAT1CISD1MAOA
SCHEMBL7768284 0.86 PTGS2 (1.00) PTGS2PTGS1NAT1CISD1GAA
Darbufelone SCHEMBL452950 0.86 PTGS2 (0.75) PTGS2PTGS1GAAALOX5
Darbufelone SCHEMBL452951 0.86 PTGS2 (0.75) PTGS2PTGS1GAAALOX5
Darbufelone SCHEMBL8526046 0.86 PTGS2 (0.75) PTGS2PTGS1GAAALOX5
SCHEMBL8618544 0.86 PTGS2 (1.00) PTGS2PTGS1NAT1CISD1GAA
SCHEMBL8309757 0.86 PTGS2 (1.00) PTGS2PTGS1NAT1CISD1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0449216-B1 3,5-di-tertiarybutyl-4-hydroxyphenylmethylene derivatives of 2-substituted thiazolidinones, oxazolidinones, and imidazolidinones as antiinflammatory agents WARNER LAMBERT CO (US) 1996-02-07 EP claimed
US-5143928-A Inhibitors of cyclooxygenase and lipoxygenase WARNER-LAMBERT COMPANY (US) 1992-09-01 US claimed
EP-0449216-A1 3,5-di-tertiarybutyl-4-hydroxyphenylmethylene derivatives of 2-substituted thiazolidinones, oxazolidinones, and imidazolidinones as antiinflammatory agents WARNER-LAMBERT COMPANY (US) 1991-10-02 EP claimed