SCHEMBL8962770

SCHEMBL8962770

N#Cc1ccc(C2CCC(CC[C@H]3CC[C@H](/C=C/Cl)CC3)CC2)cc1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 8/20 0.38
GRIA1 P42261 1/20 0.38
GRIA2 P42262 1/20 0.38
GRIA3 P42263 1/20 0.38
ESR1 P03372 6/20 0.36
CYP2C9 P11712 3/20 0.36
CYP3A4 P08684 2/20 0.36
MAOB P27338 5/20 0.35
MEN1 O00255 1/20 0.35
MAPK1 P28482 1/20 0.35
KMT2A Q03164 1/20 0.35
USP30 Q70CQ3 1/20 0.34
HSD11B1 P28845 1/20 0.34
PANK3 Q9H999 1/20 0.34
MAOA P21397 3/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8962766 1.00 ESR2 (0.38) ESR2GRIA1GRIA2GRIA3ESR1
SCHEMBL8962812 0.91 GRIA1 (0.39) GRIA1GRIA2GRIA3MAOBHSD11B1
SCHEMBL8962800 0.91 GRIA1 (0.39) GRIA1GRIA2GRIA3MAOBHSD11B1
SCHEMBL8963220 0.87 HRH3 (0.42) GRIA1GRIA2GRIA3MAOBHSD11B1
SCHEMBL8963065 0.87 GRIA1 (0.37) GRIA1GRIA2GRIA3MAOBHSD11B1
SCHEMBL8963232 0.87 HRH3 (0.42) GRIA1GRIA2GRIA3MAOBHSD11B1
SCHEMBL9510387 0.86 ESR2 (0.38) ESR2GRIA1GRIA2GRIA3ESR1
SCHEMBL8449106 0.86 ESR2 (0.38) ESR2GRIA1GRIA2GRIA3ESR1
SCHEMBL8449108 0.86 ESR2 (0.38) ESR2GRIA1GRIA2GRIA3ESR1
SCHEMBL9510390 0.86 ESR2 (0.38) ESR2GRIA1GRIA2GRIA3ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559860-B1 HALOVINYL-DERIVATIVES HOFFMANN LA ROCHE (CH) 1996-02-14 EP disclosed
US-5364556-A Halovinyl-derivatives HOFFMANN-LA ROCHE INC. (US) 1994-11-15 US disclosed