SCHEMBL8963232

SCHEMBL8963232

N#Cc1ccc(-c2ccc([C@H]3CC[C@H](/C=C/Cl)CC3)cc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.42
KCNH2 Q12809 1/20 0.42
EGLN2 Q96KS0 1/20 0.39
P2RY14 Q15391 1/20 0.39
PAX8 Q06710 1/20 0.38
HRH2 P25021 1/20 0.38
HRH1 P35367 1/20 0.38
GRIA1 P42261 1/20 0.37
GRIA2 P42262 1/20 0.37
GRIA3 P42263 1/20 0.37
MMP3 P08254 1/20 0.37
KDM1A O60341 1/20 0.37
SCD5 Q86SK9 2/20 0.36
JAK2 O60674 1/20 0.35
JAK3 P52333 1/20 0.35
PTK2 Q05397 1/20 0.35
CYP11B2 P19099 1/20 0.35
HDAC2 Q92769 1/20 0.35
MAOB P27338 2/20 0.35
KIF11 P52732 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8963220 1.00 HRH3 (0.42) HRH3KCNH2EGLN2P2RY14PAX8
SCHEMBL8962812 0.95 GRIA1 (0.39) HRH3KCNH2EGLN2GRIA1GRIA2
SCHEMBL8962800 0.95 GRIA1 (0.39) HRH3KCNH2EGLN2GRIA1GRIA2
SCHEMBL9300526 0.93 KDM1A (0.38) HRH3KCNH2EGLN2P2RY14PAX8
SCHEMBL8963065 0.91 GRIA1 (0.37) HRH3KCNH2EGLN2P2RY14GRIA1
SCHEMBL8962770 0.87 ESR2 (0.38) GRIA1GRIA2GRIA3MAOBHSD11B1
SCHEMBL8962766 0.87 ESR2 (0.38) GRIA1GRIA2GRIA3MAOBHSD11B1
SCHEMBL9475715 0.85 HRH3 (0.42) HRH3KCNH2EGLN2P2RY14PAX8
SCHEMBL9475718 0.85 HRH3 (0.42) HRH3KCNH2EGLN2P2RY14PAX8
SCHEMBL9168960 0.85 HRH3 (0.45) HRH3KCNH2EGLN2P2RY14PAX8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559860-B1 HALOVINYL-DERIVATIVES HOFFMANN LA ROCHE (CH) 1996-02-14 EP disclosed