SCHEMBL8963049

SCHEMBL8963049

O=C(O)CCc1ccc(C2CCC([C@H]3CC[C@H](/C=C/Cl)CC3)CC2)cc1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 5/20 0.40
FFAR4 Q5NUL3 8/20 0.40
HDAC2 Q92769 1/20 0.39
CYP2D6 P10635 1/20 0.39
KEAP1 Q14145 1/20 0.38
S1PR1 P21453 2/20 0.38
S1PR3 Q99500 1/20 0.38
S1PR5 Q9H228 1/20 0.38
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6488402 0.82 FFAR1 (0.57) FFAR1FFAR4CYP2D6KEAP1
SCHEMBL8963029 0.81 SPHK1 (0.43) HDAC2
SCHEMBL9408368 0.78 L3MBTL1 (0.40) FFAR4HDAC2
SCHEMBL8963210 0.78 SPHK1 (0.36) HDAC2
SCHEMBL8963144 0.76 SPHK1 (0.47) HDAC2
SCHEMBL8963157 0.76 SPHK1 (0.47) HDAC2
SCHEMBL13061403 0.76 FFAR4 (0.56) FFAR1FFAR4KEAP1S1PR1S1PR3
SCHEMBL8963019 0.75 HDAC2 (0.45) HDAC2CYP2D6
SCHEMBL8963014 0.75 HDAC2 (0.45) HDAC2CYP2D6
SCHEMBL9408347 0.75 SPHK1 (0.39) FFAR4HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559860-B1 HALOVINYL-DERIVATIVES HOFFMANN LA ROCHE (CH) 1996-02-14 EP disclosed
US-5364556-A Halovinyl-derivatives HOFFMANN-LA ROCHE INC. (US) 1994-11-15 US disclosed
WO-1993007234-A1 HALOVINYL-DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1993-04-15 WO disclosed