SCHEMBL8963198

SCHEMBL8963198

CCOc1ccc(C2CCC(CC[C@H]3CC[C@H](/C=C/Cl)CC3)CC2)cc1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.37
NQO1 P15559 1/20 0.37
ESR2 Q92731 2/20 0.36
MAPT P10636 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
MAPK1 P28482 1/20 0.36
ESR1 P03372 1/20 0.35
CYP3A4 P08684 1/20 0.35
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
RAB9A P51151 1/20 0.33
DGAT1 O75907 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8963193 1.00 CYP2C9 (0.37) CYP2C9NQO1ESR2MAPTMEN1
SCHEMBL8962983 0.93 NQO1 (0.42) CYP2C9NQO1MAPTKMT2ACYP3A4
SCHEMBL8962980 0.93 NQO1 (0.42) CYP2C9NQO1MAPTKMT2ACYP3A4
SCHEMBL8962703 0.90 RAB9A (0.39) CYP2C9ESR2MAPTMEN1KMT2A
SCHEMBL8962699 0.90 RAB9A (0.39) CYP2C9ESR2MAPTMEN1KMT2A
SCHEMBL8963401 0.89 NQO1 (0.39) CYP2C9NQO1MAPTKMT2ACYP3A4
SCHEMBL8962700 0.89 NQO1 (0.39) NQO1MAPTALDH1A1MAOAMAOB
SCHEMBL8962695 0.89 NQO1 (0.39) NQO1MAPTALDH1A1MAOAMAOB
SCHEMBL9477208 0.87 CYP2C9 (0.37) CYP2C9NQO1ESR2MAPTMEN1
SCHEMBL9477220 0.87 CYP2C9 (0.37) CYP2C9NQO1ESR2MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559860-B1 HALOVINYL-DERIVATIVES HOFFMANN LA ROCHE (CH) 1996-02-14 EP disclosed
US-5364556-A Halovinyl-derivatives HOFFMANN-LA ROCHE INC. (US) 1994-11-15 US disclosed
WO-1993007234-A1 HALOVINYL-DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1993-04-15 WO disclosed