SCHEMBL8963292

SCHEMBL8963292

Fc1cc(CC[C@H]2CC[C@H]([C@H]3CC[C@H](/C=C/Cl)CC3)CC2)ccc1Cl

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PROKR1 Q8TCW9 3/20 0.33
FPR2 P25090 2/20 0.33
KCNH2 Q12809 1/20 0.32
HTR2A P28223 2/20 0.31
HTR2C P28335 2/20 0.31
TRPA1 O75762 1/20 0.31
PTGIR P43119 1/20 0.31
PTGDR Q13258 1/20 0.31
MAPK1 P28482 1/20 0.31
RPS6KA1 Q15418 1/20 0.31
DRD4 P21917 1/20 0.30
SIGMAR1 Q99720 1/20 0.30
MAOA P21397 1/20 0.30
MAOB P27338 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8963287 1.00 PROKR1 (0.33) PROKR1FPR2KCNH2HTR2AHTR2C
SCHEMBL8963053 0.96 KCNH2 (0.33) PROKR1FPR2KCNH2TRPA1PTGIR
SCHEMBL8963047 0.96 KCNH2 (0.33) PROKR1FPR2KCNH2TRPA1PTGIR
SCHEMBL9540834 0.89 GRM2 (0.32) PROKR1FPR2KCNH2
SCHEMBL9265780 0.89 PROKR1 (0.35) PROKR1FPR2KCNH2HTR2AHTR2C
SCHEMBL9265765 0.89 PROKR1 (0.35) PROKR1FPR2KCNH2HTR2AHTR2C
SCHEMBL9265783 0.89 PROKR1 (0.35) PROKR1FPR2KCNH2HTR2AHTR2C
SCHEMBL9265771 0.89 PROKR1 (0.35) PROKR1FPR2KCNH2HTR2AHTR2C
SCHEMBL9450833 0.86 CNR1 (0.32)
SCHEMBL9255736 0.86 PROKR1 (0.34) PROKR1FPR2KCNH2HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559860-B1 HALOVINYL-DERIVATIVES HOFFMANN LA ROCHE (CH) 1996-02-14 EP disclosed
US-5364556-A Halovinyl-derivatives HOFFMANN-LA ROCHE INC. (US) 1994-11-15 US disclosed
EP-0559860-A1 HALOVINYL-DERIVATIVES. HOFFMANN LA ROCHE (CH) 1993-09-15 EP disclosed
WO-1993007234-A1 HALOVINYL-DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1993-04-15 WO disclosed