SCHEMBL8964561

SCHEMBL8964561

COc1cc2c(cc1OCc1ccccc1)C[C@@H](C(=O)O)NC2

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 1/20 0.54
PDE4B Q07343 2/20 0.50
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
PKM P14618 1/20 0.48
SRD5A1 P18405 2/20 0.48
SRD5A2 P31213 2/20 0.48
CHRNA7 P36544 2/20 0.47
HPGD P15428 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
PDE4A P27815 1/20 0.46
PDE4C Q08493 1/20 0.46
PDE4D Q08499 1/20 0.46
SMPD1 P17405 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8964158 1.00 AGTR2 (0.54) AGTR2PDE4BNPC1RAB9APKM
SCHEMBL243337 0.91 AGTR2 (0.50) AGTR2PDE4BNPC1RAB9APKM
SCHEMBL1202600 0.85 EGLN1 (0.44)
SCHEMBL4464347 0.85 EGLN1 (0.44)
SCHEMBL7225047 0.85 ACE (0.47) AGTR2PDE4BNPC1RAB9APKM
SCHEMBL7225043 0.85 ACE (0.47) AGTR2PDE4BNPC1RAB9APKM
Hydrochloric Acid SCHEMBL7221546 0.84 EGLN1 (0.43) HDAC8
Hydrochloric Acid SCHEMBL7221540 0.84 EGLN1 (0.43) HDAC8
SCHEMBL3054428 0.83 CHRNA7 (0.51) AGTR2PDE4BCHRNA7PDE4APDE4C
SCHEMBL3051394 0.82 CHRNA7 (0.50) AGTR2PDE4BNPC1RAB9ACHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5525614-A TREATING VASCULAR RESTENOSIS, CNS DISORDERS WARNER-LAMBERT COMPANY (US) 1996-06-11 US disclosed
US-5489686-A CARDIOVASCULAR DISORDER, NERVOUS SYSTEM DISORDER, ANTIDIURETIC , PSYCHLOGICAL DISORDER, ANTIDEPRESSANTS WARNER-LAMBERT COMPANY (US) 1996-02-06 US disclosed
US-5350757-A Treatment of vascular restenosis, nervous system disorders and cognition enhancement WARNER-LAMBERT COMPANY (US) 1994-09-27 US disclosed
US-5246943-A Substituted 1,2,3,4-tetahydroisoquinolines with angiotensin II receptor antagonist properties WARNER-LAMBERT COMPANY (US) 1993-09-21 US disclosed