SCHEMBL8964661

SCHEMBL8964661

C=CCc1cc(Cl)sc1Cl

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.39
GABRA1 P14867 2/20 0.36
GABRB2 P47870 2/20 0.36
GSK3B P49841 1/20 0.35
DAO P14920 1/20 0.34
PTGDR Q13258 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
GRIA1 P42261 2/20 0.32
GRIA2 P42262 2/20 0.32
GRIA3 P42263 2/20 0.32
GRIA4 P48058 2/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16703534 0.81 GABRA1 (0.33) GABRA1GABRB2PTGDRPTGDR2
SCHEMBL16703569 0.81 GABRA1 (0.33) GABRA1GABRB2PTGDRPTGDR2
SCHEMBL12987883 0.79 GABRA1 (0.36) GAAGABRA1GABRB2GSK3BPTGDR
SCHEMBL6184676 0.77 GSK3B (0.39) GSK3BDAO
SCHEMBL11766536 0.69 GABRA1 (0.40) GAAGABRA1GABRB2PTGDRPTGDR2
SCHEMBL843790 0.69
SCHEMBL44699 0.68 GABRA1 (0.48) GAAGABRA1GABRB2POLB
SCHEMBL29259237 0.67
SCHEMBL16235099 0.65 CYP1A2 (0.36) GSK3BDAO
SCHEMBL12362660 0.65 GSK3B (0.36) GSK3BDAOGRIA1GRIA2GRIA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015070028-A2 METHOD OF SYNTHESIS OF POLYTHIOPHENES OF CONTROLLED MOLECULAR WEIGHT RIEKE REUBEN (US) 2015-05-14 WO disclosed
EP-0410379-B1 Pharmaceutically active 3-aryl and 3-heteroaryl-2-fluoro-1-olefins MERRELL DOW PHARMA (US) 1996-01-31 EP disclosed
US-5068465-A Hypotensive agents or enzyme inhibitors for treatment of hypertension MERRELL DOW PHARMACEUTICALS INC. (US) 1991-11-26 US disclosed
EP-0410379-A2 Pharmaceutically active 3-aryl and 3-heteroaryl-2-fluoro-1-olefins MERRELL DOW PHARMACEUTICALS INC. (US) 1991-01-30 EP disclosed
US-4981868-A ENZYME INHIBITORS, HYPOTENSIVES MERRELL DOW PHARMACEUTICAL (US) 1991-01-01 US disclosed