SCHEMBL8964774

SCHEMBL8964774

C=C(F)Cc1ccc(Br)s1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
KDM4E B2RXH2 4/20 0.38
ALDH1A1 P00352 3/20 0.38
TDP1 Q9NUW8 3/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
CES2 O00748 1/20 0.35
CES1 P23141 1/20 0.35
GSK3B P49841 2/20 0.35
DAO P14920 1/20 0.34
GAA P10253 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
ESR1 P03372 1/20 0.31
AR P10275 1/20 0.31
MAPT P10636 1/20 0.30
HTT P42858 1/20 0.30
PARP1 P09874 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8964660 0.74 PRMT6 (0.47) KDM4EALDH1A1L3MBTL1DAOGAA
SCHEMBL9699843 0.72 GSK3B (0.46) HDAC1HDAC6KDM4EALDH1A1TDP1
SCHEMBL29242041 0.72
SCHEMBL1414863 0.71 KDM4E (0.45) HDAC1HDAC6KDM4EALDH1A1TDP1
SCHEMBL13049960 0.71 KDM4E (0.45) HDAC1HDAC6KDM4EALDH1A1TDP1
SCHEMBL1522719 0.69
SCHEMBL13873989 0.69
SCHEMBL1598343 0.68 HDAC1 (0.44) HDAC1HDAC6KDM4ETDP1L3MBTL1
SCHEMBL8773498 0.67
SCHEMBL223822 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0410379-B1 Pharmaceutically active 3-aryl and 3-heteroaryl-2-fluoro-1-olefins MERRELL DOW PHARMA (US) 1996-01-31 EP disclosed