SCHEMBL8965502

SCHEMBL8965502

NC(COCc1cccc(Br)c1)C(c1ccccc1)c1ccccc1

nearest known ligand 0.79

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 17/20 0.79
IDO1 P14902 2/20 0.49
AGXT P21549 2/20 0.49
MAOB P27338 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8965500 0.88 TACR1 (1.00) TACR1
SCHEMBL8965434 0.85 TACR1 (1.00) TACR1
SCHEMBL8966079 0.83 TACR1 (1.00) TACR1IDO1AGXT
SCHEMBL8965360 0.82 TACR1 (1.00) TACR1
SCHEMBL8965741 0.80 TACR1 (0.67) TACR1
SCHEMBL8965336 0.79 TACR1 (1.00) TACR1
SCHEMBL7965713 0.79 IDO1 (0.54) TACR1IDO1AGXTMAOB
SCHEMBL7965716 0.79 IDO1 (0.54) TACR1IDO1AGXTMAOB
SCHEMBL8965372 0.78 TACR1 (0.63) TACR1
SCHEMBL8912140 0.77 TACR1 (1.00) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0593557-B1 AROMATIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY MERCK SHARP & DOHME (GB) 1996-01-31 EP claimed
EP-0593557-A1 AROMATIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY. MERCK SHARP & DOHME (GB) 1994-04-27 EP claimed
WO-1993001160-A1 AROMATIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY MERCK SHARP & DOHME LIMITED (GB) 1993-01-21 WO claimed
EP-0522808-A2 Aromatic compounds, pharmaceutical compositions containing them and their use in therapy MERCK SHARP & DOHME LTD. (GB) 1993-01-13 EP claimed