SCHEMBL8965741

SCHEMBL8965741

N#Cc1cccc(COCC(N)C(c2ccccc2)c2ccccc2)c1

nearest known ligand 0.67

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 16/20 0.67
MRGPRX1 Q96LB2 1/20 0.45
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
FFAR1 O14842 1/20 0.41
FFAR4 Q5NUL3 1/20 0.41
MRGPRX4 Q96LA9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8965434 0.81 TACR1 (1.00) TACR1
SCHEMBL8966079 0.80 TACR1 (1.00) TACR1
SCHEMBL8965502 0.80 TACR1 (0.79) TACR1
SCHEMBL31568453 0.78 TSHR (0.56) TACR1MRGPRX1SLC6A2SLC6A4FFAR1
SCHEMBL22469683 0.78 TSHR (0.56) TACR1MRGPRX1SLC6A2SLC6A4FFAR1
SCHEMBL6668868 0.76 MRGPRX4 (0.55) SLC6A4FFAR1FFAR4MRGPRX4
SCHEMBL8965372 0.74 TACR1 (0.63) TACR1
SCHEMBL28384912 0.74 MRGPRX4 (0.50) FFAR1FFAR4MRGPRX4
SCHEMBL8965500 0.73 TACR1 (1.00) TACR1
SCHEMBL8912140 0.73 TACR1 (1.00) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0593557-B1 AROMATIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY MERCK SHARP & DOHME (GB) 1996-01-31 EP claimed
WO-1993001160-A1 AROMATIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY MERCK SHARP & DOHME LIMITED (GB) 1993-01-21 WO claimed
EP-0522808-A2 Aromatic compounds, pharmaceutical compositions containing them and their use in therapy MERCK SHARP & DOHME LTD. (GB) 1993-01-13 EP claimed