SCHEMBL8965617

SCHEMBL8965617

Cc1ccc(C)c(COc2ccc(N)nn2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.41
ALDH1A1 P00352 5/20 0.40
HPGD P15428 4/20 0.40
TACR1 P25103 1/20 0.38
HTT P42858 3/20 0.36
KDM4E B2RXH2 2/20 0.36
POLB P06746 1/20 0.36
BCAT2 O15382 1/20 0.36
ABL1 P00519 1/20 0.35
SRC P12931 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
CYP19A1 P11511 1/20 0.34
NOS3 P29474 2/20 0.34
NOS2 P35228 2/20 0.34
MAPT P10636 1/20 0.34
NCK1 P16333 1/20 0.33
BACE1 P56817 1/20 0.33
MEN1 O00255 1/20 0.33
NOS1 P29475 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8965946 0.76 IDO1 (0.51) TAAR1ALDH1A1TDP1
SCHEMBL8965867 0.75 FFAR1 (0.38) ALDH1A1HTTPOLBBCAT2NOS3
SCHEMBL8966010 0.75 BCAT2 (0.45) ALDH1A1HPGDHTTKDM4EBCAT2
SCHEMBL3968418 0.71 TAAR1 (0.50) TAAR1ALDH1A1TACR1POLBABL1
SCHEMBL3109560 0.71 KDM4C (0.41) ALDH1A1HPGDHTTKDM4EPOLB
SCHEMBL4023051 0.70 KMT2A (0.49) ALDH1A1BCAT2TDP1MAPTNCK1
Hydrochloric Acid SCHEMBL6364077 0.70 TAAR1 (0.49) TAAR1ALDH1A1TACR1POLBABL1
SCHEMBL8965974 0.70 IDO1 (0.51) TAAR1ALDH1A1POLBBCAT2MAPT
SCHEMBL13929700 0.70 NPC1 (0.47) TAAR1TACR1ABL1SRCTDP1
SCHEMBL2349832 0.69 BCAT2 (0.47) ALDH1A1HPGDHTTKDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5538970-A Treatment of cancer with imidazo-1,2-pyridazin compounds GLAXO WELLCOME INC. (US) 1996-07-23 US disclosed
US-5447956-A Anticarcinogenic agents BURROUGHS WELLCOME CO. (US) 1995-09-05 US disclosed
US-5380759-A Methyl N-[6-(3,4,5-trimethoxybenzloxy)imidazo[1,2-b]pyridazin-2-zyl]carbamate used to treat leukemia BURROUGHS WELLCOME CO. (US) 1995-01-10 US disclosed
US-5371219-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1994-12-06 US disclosed
EP-0305093-B1 Imidazo(1,2-b)pyridazine derivatives WELLCOME FOUND (GB) 1994-04-06 EP disclosed
US-5091531-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1992-02-25 US disclosed
EP-0305093-A1 Imidazo(1,2-b)pyridazine derivatives THE WELLCOME FOUNDATION LIMITED (GB) 1989-03-01 EP disclosed