SCHEMBL8965802

SCHEMBL8965802

Brc1ccc(C2c3ccccc3-c3ccc4ccccc4c32)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
NPC1 O15118 1/20 0.44
GAA P10253 1/20 0.44
POLB P06746 2/20 0.43
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40
KLK3 P07288 1/20 0.39
AR P10275 1/20 0.39
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
HTT P42858 1/20 0.34
RECQL P46063 1/20 0.34
CYP1A1 P04798 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP1B1 Q16678 1/20 0.34
KDM1A O60341 2/20 0.33
RCOR1 Q9UKL0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8966049 0.87 ESR1 (0.41) TP53MAPTESR1ESR2AR
SCHEMBL17765439 0.81 HPGD (0.48) MEN1KMT2ANPC1GAATP53
SCHEMBL17777815 0.81 ESR1 (0.39) MEN1KMT2AGAAPOLBMAPT
SCHEMBL7520996 0.78 KMT2A (0.61) MEN1KMT2ANPC1GAAALDH1A1
Benzene SCHEMBL28134446 0.76 MEN1 (0.59) MEN1KMT2ANPC1GAATP53
SCHEMBL28081301 0.76 KMT2A (0.44) MEN1KMT2ANPC1GAAALDH1A1
SCHEMBL27880163 0.75 KMT2A (0.46) MEN1KMT2ANPC1GAATP53
SCHEMBL27967593 0.74 KMT2A (0.45) MEN1KMT2ANPC1GAAALDH1A1
SCHEMBL10685337 0.74 KDM1A (0.42) NPC1MAPTESR1ESR2ALDH1A1
SCHEMBL18926276 0.73 NPC1 (0.55) MEN1KMT2ANPC1GAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0524742-B1 Benzo(a)fluorene compounds LILLY CO ELI (US) 1996-02-28 EP disclosed
EP-0524742-A2 Benzo(a)fluorene compounds ELI LILLY AND COMPANY (US) 1993-01-27 EP disclosed
US-5147880-A Estrogenic and antiestrogenic activity ELI LILLY AND COMPANY (US) 1992-09-15 US disclosed