SCHEMBL10685337

SCHEMBL10685337

NC1c2ccccc2-c2ccc3ccccc3c21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.42
ALDH1A1 P00352 6/20 0.39
HSD17B10 Q99714 3/20 0.39
TSHR P16473 2/20 0.39
CYP2A6 P11509 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
DNMT1 P26358 1/20 0.38
HPRT1 P00492 1/20 0.37
HTR7 P34969 2/20 0.36
HTR2B P41595 2/20 0.36
HTR2A P28223 1/20 0.35
KDM4E B2RXH2 3/20 0.35
MAPT P10636 2/20 0.35
HPGD P15428 2/20 0.35
MAPK1 P28482 2/20 0.35
TDP2 O95551 1/20 0.35
ALOX12 P18054 1/20 0.35
CASP3 P42574 1/20 0.35
HTT P42858 1/20 0.35
GALK1 P51570 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24023063 0.80 KDM1A (0.38) KDM1AALDH1A1HSD17B10TSHRCYP2A6
SCHEMBL8966049 0.79 ESR1 (0.41) KDM1AALDH1A1HSD17B10TSHRCYP2A6
SCHEMBL29941360 0.78 HPRT1 (0.50) KDM1AALDH1A1HSD17B10TSHRCYP2A6
SCHEMBL1897664 0.78 KDM1A (0.48) KDM1AALDH1A1HSD17B10TSHRCYP2A6
Hydrochloric Acid SCHEMBL4832739 0.78 ALDH1A1 (0.39) KDM1AALDH1A1HSD17B10TSHRCYP2A6
SCHEMBL5999291 0.78 ALDH1A1 (0.40) ALDH1A1HSD17B10TSHRCYP2A6TDP1
SCHEMBL9123563 0.74 HDAC3 (0.36) KDM1AALDH1A1HSD17B10TSHRCYP2A6
SCHEMBL8965802 0.74 MEN1 (0.44) KDM1AALDH1A1HSD17B10TSHRCYP2A6
SCHEMBL16671741 0.73 HPRT1 (0.35) KDM1AALDH1A1HSD17B10TSHRTDP1
SCHEMBL29444048 0.72 HTR2A (0.52) KDM1AALDH1A1HTR7HTR2BHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 359 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4426701-B1 BENZOFURO[3,2-D]PYRIMIDIN-2,4-DICARBONITRILE DERIVATIVES AND SIMILAR COMPOUNDS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2026-05-20 EP disclosed
EP-4242286-B1 MATERIALS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2026-04-29 EP disclosed
EP-4441048-B1 TRIPHENYLENE-TRIAZINE-DIBENZOFURANE/DIBENZOTHIOPHENE DERIVATIVES FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2026-04-22 EP disclosed
EP-4724542-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES Merck Patent GmbH (DE) 2026-04-15 EP disclosed
EP-4078692-B1 COMPOUNDS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2026-03-18 EP disclosed
WO-2025228800-A1 MATERIALS FOR ORGANIC ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2025-11-06 WO disclosed
EP-4638439-A1 NOVEL MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES Merck Patent GmbH (DE) 2025-10-29 EP disclosed
EP-4410073-B1 ORGANIC ELECTROLUMINESCENT APPARATUS MERCK PATENT GMBH (DE) 2025-10-29 EP disclosed
EP-4410072-B1 ORGANIC ELECTROLUMINESCENT APPARATUS MERCK PATENT GMBH (DE) 2025-10-29 EP disclosed
EP-4634166-A1 MATERIALS FOR ELECTRONIC DEVICES Merck Patent GmbH (DE) 2025-10-22 EP disclosed
EP-2907173-A1 ELECTRONIC DEVICE Merck Patent GmbH (DE) 2015-08-19 EP disclosed
WO-2015049022-A1 TRIARYLAMINE-SUBSTITUTED BENZO[H]QUINOLINE-DERIVATIVES AS MATERIALS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2015-04-09 WO disclosed
WO-2015022051-A1 MATERIALS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2015-02-19 WO disclosed
WO-2015000549-A1 MATERIALS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2015-01-08 WO disclosed
WO-2014111269-A2 MATERIALS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2014-07-24 WO disclosed
WO-2014079527-A1 MATERIALS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2014-05-30 WO disclosed
WO-2014067614-A1 ELECTRONIC DEVICE MERCK PATENT GMBH (DE) 2014-05-08 WO disclosed
US-4766110-A INHIBITS ANGIOTENSIN CONVERTING ENZYME, HYPOTENSIVE AGENTS RYAN JAMES W (US) 1988-08-23 US disclosed
EP-0073143-B1 NOVEL COMPLEX AMIDO AND IMIDO DERIVATIVES OF CARBOXYALKYL PEPTIDES AND THIOETHERS AND ETHERS OF PEPTIDES Ryan, James Walter (US) 1985-11-21 EP disclosed
EP-0073143-A2 Novel complex amido and imido derivatives of carboxyalkyl peptides and thioethers and ethers of peptides Ryan, James Walter (US) 1983-03-02 EP disclosed