SCHEMBL8965933

SCHEMBL8965933

COC(=O)Nc1cn2nc(OCc3ccccc3C(C)(C)C)ccc2n1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.40
CSNK1D P48730 1/20 0.39
RIPK1 Q13546 13/20 0.38
PIK3CA P42336 1/20 0.37
PDE10A Q9Y233 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9157347 0.91 PDE10A (0.41) KDRCSNK1DRIPK1PIK3CAPDE10A
SCHEMBL8965615 0.88 RIPK1 (0.41) KDRCSNK1DRIPK1PIK3CAPDE10A
SCHEMBL8965537 0.86 RIPK1 (0.43) KDRCSNK1DRIPK1PIK3CA
SCHEMBL8965637 0.85 ATM (0.44) KDRCSNK1DRIPK1PIK3CAPDE10A
SCHEMBL8966250 0.84 CSNK1D (0.39) KDRCSNK1DRIPK1PIK3CAPDE10A
SCHEMBL9280653 0.84 CSNK1D (0.44) CSNK1DRIPK1PIK3CAPDE10A
SCHEMBL8966017 0.81 KDR (0.41) KDRCSNK1DRIPK1PIK3CA
SCHEMBL8965870 0.81 PDE10A (0.42) KDRCSNK1DPIK3CAPDE10A
SCHEMBL8965899 0.79 KDR (0.40) KDRCSNK1DRIPK1PIK3CA
SCHEMBL8965955 0.79 KDR (0.43) KDRPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5538970-A Treatment of cancer with imidazo-1,2-pyridazin compounds GLAXO WELLCOME INC. (US) 1996-07-23 US disclosed
US-5447956-A Anticarcinogenic agents BURROUGHS WELLCOME CO. (US) 1995-09-05 US disclosed
US-5371219-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1994-12-06 US disclosed