SCHEMBL8967589

SCHEMBL8967589

O=CNc1cccc(-c2ccccc2)c1

nearest known ligand 0.64

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.64
MGLL Q99685 2/20 0.55
DHODH Q02127 2/20 0.49
CA2 P00918 1/20 0.47
FDPS P14324 1/20 0.47
MMP8 P22894 1/20 0.47
MMP14 P50281 1/20 0.47
CA9 Q16790 1/20 0.47
CA14 Q9ULX7 1/20 0.47
POLB P06746 2/20 0.46
CNR1 P21554 3/20 0.45
LIMK1 P53667 1/20 0.44
SIRT2 Q8IXJ6 1/20 0.44
SIRT1 Q96EB6 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28214132 0.96 ALDH1A1 (0.56) ALDH1A1MGLLDHODHCA2FDPS
SCHEMBL27895559 0.89 ALDH1A1 (0.65) ALDH1A1MGLLDHODHCA2FDPS
SCHEMBL14471626 0.85 ALDH1A1 (0.60) ALDH1A1MGLLDHODHCA2FDPS
SCHEMBL28254478 0.85 ALDH1A1 (0.60) ALDH1A1MGLLDHODHCA2FDPS
SCHEMBL11194081 0.85 CNR1 (0.50) ALDH1A1MGLLDHODHCNR1LIMK1
SCHEMBL4429931 0.84 TRIM24 (0.59) ALDH1A1MGLLMEN1KMT2A
SCHEMBL12129057 0.82 ALDH1A1 (0.67) ALDH1A1LIMK1MEN1KMT2A
SCHEMBL18654163 0.81 HDAC6 (0.60) ALDH1A1LIMK1MEN1KMT2A
SCHEMBL223423 0.80 ALDH1A1 (0.73) ALDH1A1MGLLDHODHMMP8MMP14
SCHEMBL14418354 0.80 ALDH1A1 (0.73) ALDH1A1MGLLDHODHMMP8MMP14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108883122-A C-glycoside compounds useful for the treatment of diseases 菲姆布里昂医疗公司 2018-11-23 CN claimed
CN-108778288-A It can be used for treating antagonist derived from the mannose of the FimH of disease 菲姆布里昂医疗公司 2018-11-09 CN claimed
CN-108883122-A C-glycoside compounds useful for the treatment of diseases 菲姆布里昂医疗公司 2018-11-23 CN disclosed
CN-108778288-A It can be used for treating antagonist derived from the mannose of the FimH of disease 菲姆布里昂医疗公司 2018-11-09 CN disclosed
CN-107922394-A 3 tetrazole radical benzene, 1,2 disulfonic acid amide derivative as metal beta lactamase restrainer 默沙东公司 2018-04-17 CN disclosed
CN-104903300-B COMT inhibitor 霍夫曼-拉罗奇有限公司 2018-04-17 CN disclosed
CN-105102449-B Antiviral compound 豪夫迈·罗氏有限公司 2017-06-13 CN disclosed
CN-103442566-A Compounds for treatment of cancer GTX INC 2013-12-11 CN disclosed
CN-102883607-A Compounds for the treatment of cancer GTX INC (US) 2013-01-16 CN disclosed
EP-2543437-A2 HOMOGENEOUS ASYMMETRIC HYDROGENATION CATALYST Takasago International Corporation (JP) 2013-01-09 EP disclosed
CN-102746285-A Compounds and compositions as HEDGEHOG pathway modulators IRM LLC 2012-10-24 CN disclosed
CN-102170873-A Smoothied antagonism for treating disorders associated with HEDGEHOG pathways NOVARTIS AG 2011-08-31 CN disclosed
US-5530138-A A PYRROLIZINE DERIVATIVE; EFFECTIVE IN THE TREATMENT OF SENILE DEMENTIA SANWA KAGAKU KENKYUSHO CO., LTD. (JP) 1996-06-25 US disclosed
EP-0647642-A1 1-Azabicyclo(3.3.0)octane derivatives and their use SANWA KAGAKU KENKYUSHO CO., LTD. (JP) 1995-04-12 EP disclosed